Direct Synthesis of Azaheterocycles from N-Aryl/Vinyl Amides. Synthesis of 4-(Methylthio)-2-phenylquinazoline and 4-(4-Methoxyphenyl)-2-phenylquinoline
A flame-dried, 300-mL three-necked round-bottomed flask equipped with a 3.0 cm footballshaped stir bar, rubber septum, and low temperature thermometer is charged with benzanilide (1) (Note 1) (6.02 g, 30.5 mmol, 1 equiv), sealed under an argon atmosphere, and fitted with an argon inlet. Anhydrous di...
Main Authors: | Kaise, Hiromi, Movassaghi, Mohammad, Ahmad, Omar K., Medley, Jonathan William, Coste, Alexis |
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Other Authors: | Massachusetts Institute of Technology. Department of Chemistry |
Format: | Article |
Published: |
Organic Syntheses, Inc.
2018
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Online Access: | http://hdl.handle.net/1721.1/114182 https://orcid.org/0000-0003-3080-1063 |
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