Efficient Pd-Catalyzed Amination Reactions for Heterocycle Functionalization
The Pd-catalyzed amination of unprotected benzo-fused heterocycles is reported, which allows for greater flexibility and efficiency in the modification of this important class of molecules. The generality of these simple and efficient procedures is demonstrated through the synthesis of a wide variet...
Main Authors: | Henderson, Jaclyn L., Buchwald, Stephen Leffler |
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Other Authors: | Massachusetts Institute of Technology. Department of Chemistry |
Format: | Article |
Language: | en_US |
Published: |
Organic Letters
2012
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Online Access: | http://hdl.handle.net/1721.1/71942 https://orcid.org/0000-0003-3875-4775 |
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