Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids
A palladium-catalyzed method for the preparation of sulfonamides is described. The process exhibits significant functional group tolerance and allows for the preparation of a number of arylsulfonyl chlorides and sulfonamides under mild conditions.
| Main Authors: | , , |
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| Other Authors: | |
| Format: | Article |
| Language: | en_US |
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American Chemical Society (ACS)
2015
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| Online Access: | http://hdl.handle.net/1721.1/93910 https://orcid.org/0000-0003-3875-4775 |
| _version_ | 1826206354944032768 |
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| author | Niljianskul, Nootaree DeBergh, John Robbins Buchwald, Stephen Leffler |
| author2 | Massachusetts Institute of Technology. Department of Chemistry |
| author_facet | Massachusetts Institute of Technology. Department of Chemistry Niljianskul, Nootaree DeBergh, John Robbins Buchwald, Stephen Leffler |
| author_sort | Niljianskul, Nootaree |
| collection | MIT |
| description | A palladium-catalyzed method for the preparation of sulfonamides is described. The process exhibits significant functional group tolerance and allows for the preparation of a number of arylsulfonyl chlorides and sulfonamides under mild conditions. |
| first_indexed | 2024-09-23T13:27:51Z |
| format | Article |
| id | mit-1721.1/93910 |
| institution | Massachusetts Institute of Technology |
| language | en_US |
| last_indexed | 2024-09-23T13:27:51Z |
| publishDate | 2015 |
| publisher | American Chemical Society (ACS) |
| record_format | dspace |
| spelling | mit-1721.1/939102022-10-01T15:26:56Z Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids Niljianskul, Nootaree DeBergh, John Robbins Buchwald, Stephen Leffler Massachusetts Institute of Technology. Department of Chemistry DeBergh, John Robbins Niljianskul, Nootaree Buchwald, Stephen Leffler A palladium-catalyzed method for the preparation of sulfonamides is described. The process exhibits significant functional group tolerance and allows for the preparation of a number of arylsulfonyl chlorides and sulfonamides under mild conditions. National Institutes of Health (U.S.) (GM58160) National Institutes of Health (U.S.) (Fellowship 1F32GM099202) 2015-02-06T19:43:46Z 2015-02-06T19:43:46Z 2013-07 2013-06 Article http://purl.org/eprint/type/JournalArticle 0002-7863 1520-5126 http://hdl.handle.net/1721.1/93910 DeBergh, J. Robb, Nootaree Niljianskul, and Stephen L. Buchwald. “Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids.” Journal of the American Chemical Society 135, no. 29 (July 24, 2013): 10638–10641. https://orcid.org/0000-0003-3875-4775 en_US http://dx.doi.org/10.1021/ja405949a Journal of the American Chemical Society Article is made available in accordance with the publisher's policy and may be subject to US copyright law. Please refer to the publisher's site for terms of use. application/pdf American Chemical Society (ACS) PMC |
| spellingShingle | Niljianskul, Nootaree DeBergh, John Robbins Buchwald, Stephen Leffler Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids |
| title | Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids |
| title_full | Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids |
| title_fullStr | Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids |
| title_full_unstemmed | Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids |
| title_short | Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids |
| title_sort | synthesis of aryl sulfonamides via palladium catalyzed chlorosulfonylation of arylboronic acids |
| url | http://hdl.handle.net/1721.1/93910 https://orcid.org/0000-0003-3875-4775 |
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