Biomass derived furfural-based facile synthesis of protected (2S)-phenyl-3-piperidone, a common intermediate for many drugs
An efficient synthetic route towards tosyl-protected (2S)-phenyl-3-piperidone, a common intermediate for many drugs, has been developed in 5 steps in 54% yield from biomass derived furfural. The synthetic utility of the piperidone core structure was demonstrated with the synthesis of a NK1 receptor...
Hlavní autoři: | , , , |
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Další autoři: | |
Médium: | Journal Article |
Jazyk: | English |
Vydáno: |
2015
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Témata: | |
On-line přístup: | https://hdl.handle.net/10356/79354 http://hdl.handle.net/10220/25021 |