A tandem Heck–aza-Michael addition protocol for the one-pot synthesis of isoindolines from unprotected amines

A tandem Heck–aza-Michael addition protocol for the one-pot synthesis of isoindolines from unprotected amines

A palladacycle-catalyzed tandem Heck-intramolecular aza-Michael reaction protocol has been developed for the one-pot synthesis of 1-substituted isoindolines from N-unprotected 2-bromobenzylamines and acrylates with high yields.

书目详细资料
Main Authors:	Chen, Ke, Pullarkat, Sumod A.
其他作者:	School of Physical and Mathematical Sciences
格式:	Journal Article
语言:	English
出版:	2013
主题:	DRNTU::Science::Chemistry::Organic chemistry
在线阅读:	https://hdl.handle.net/10356/99176 http://hdl.handle.net/10220/17155

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