S32212, a novel serotonin type 2C receptor inverse agonist/α2-adrenoceptor antagonist and potential antidepressant: II. A behavioral, neurochemical, and electrophysiological characterization.

S32212, a novel serotonin type 2C receptor inverse agonist/α2-adrenoceptor antagonist and potential antidepressant: II. A behavioral, neurochemical, and electrophysiological characterization.

The present studies characterized the functional profile of N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-1,2-dihydro-3-H-benzo[e]indole-3-carboxamide) (S32212), a combined serotonin (5-HT)(2C) receptor inverse agonist and α(2)-adrenoceptor antagonist that also possesses 5-HT(2A) antagonist propert...

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Bibliographic Details
Main Authors:	Dekeyne, A, Brocco, M, Loiseau, F, Gobert, A, Rivet, J, Di Cara, B, Cremers, T, Flik, G, Fone, K, Watson, D, Papp, M, Sharp, T, Serres, F, Cespuglio, R, Olivier, B, Chan, J, Lavielle, G, Millan, M
Format:	Journal article
Language:	English
Published:	2012

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