A fluorescent benzo[g]isoquinoline-based HIF prolyl hydroxylase inhibitor for cellular imaging

A fluorescent benzo[g]isoquinoline-based HIF prolyl hydroxylase inhibitor for cellular imaging

Prolyl hydroxylation domain (PHD) enzymes catalyze the hydroxylation of the transcription factor hypoxia‐inducible factor (HIF) and serve as cellular oxygen sensors. HIF and the PHD enzymes regulate numerous potentially tissue‐protective target genes which can adapt cells to metabolic and ischemic s...

Disgrifiad llawn

Manylion Llyfryddiaeth
Prif Awduron:	Mayer, M, Fey, K, Heinze, E, Rainer Wick, C, Abboud, M, Yeh, T, Tumber, A, Orth, N, Schley, G, Buchholz, B, Clark, T, Schofield, C, Willam, C, Burzlaff, N
Fformat:	Journal article
Cyhoeddwyd:	Wiley 2018

Eitemau Tebyg

No benefit of HIF prolyl hydroxylase inhibition for hypertensive renal damage in renovascular hypertensive rats
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Cyhoeddwyd: (2023-06-01)

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Cyhoeddwyd: (2016)

Molecular and Cellular Mechanisms of HIF Prolyl Hydroxylase inhibitors in Clinical Trials
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Cyhoeddwyd: (2019)

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Cyhoeddwyd: (2019)

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Cyhoeddwyd: (2010)

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Cyhoeddwyd: (2004)

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Cyhoeddwyd: (2005)

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Cyhoeddwyd: (2007)

Structural, biochemical and inhibition studies on hypoxia-inducible factor (HIF) prolyl hydroxylases
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Cyhoeddwyd: (2018)

Impact of HIF prolyl hydroxylase inhibitors in heart failure patients with renal anemia
gan: Takahiro Kambara, et al.
Cyhoeddwyd: (2024-03-01)