PURINES, PYRIMIDINES, AND IMIDAZOLES .53. SYNTHESIS OF SOME 5-HALOGENO-ANALOGUES OF METIAMIDE AND CIMETIDINE
Ethyl 5-chloroimidazole-4-carboxylate has been prepared by diazotisation of ethyl 5-amino-1-(di-O-isopropylidene-α- or -α,β-D- mannofuranosyl)imidazole-4-carboxylate, reaction of the diazonium salt with copper(I) chloride and removal of the 1-substituent with hydrochloric acid, or by similar convers...
| Main Authors: | , , |
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| Format: | Journal article |
| Language: | English |
| Published: |
1980
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