Synthetic access to 3,4-disubstituted pyroglutamates from tetramate derivatives from serine, allo-threonine and cysteine
A route allowing the conversion of substituted tetramates to 3,4-disubstituted pyroglutamates, making use of Suzuki coupling on an enol mesylate, followed by reduction, is both general and fully stereoselective.
Podrobná bibliografie
| Hlavní autoři: |
Bagum, H,
Christensen, KE,
Genov, M,
Pretsch, A,
Pretsch, D,
Moloney, MG |
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| Médium: | Journal article
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| Jazyk: | English |
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| Vydáno: |
Elsevier
2019
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