Enantio- and diastereoselective catalytic alkylation reactions with aziridines.
The first asymmetric phase transfer catalyzed alkylation reaction of a range of carbon acids with N-sulfonyl aziridines is reported. When 10 mol % of a cinchona derived quaternary ammonium salt was employed as the catalyst under mildly basic conditions, N-o-(trifluoromethane)benzenesulfonyl aziridin...
Main Authors: | , , |
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格式: | Journal article |
语言: | English |
出版: |
2008
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