Highly functionalized terpyridines as competitive inhibitors of AKAP-PKA interactions.
A good fit: Interactions between A-kinase anchoring proteins (AKAPs) and protein kinaseA (PKA) play key roles in a plethora of physiologically relevant processes whose dysregulation causes or is associated with diseases such as heart failure. Terpyridines have been developed as α-helix mimetics for...
Main Authors: | Schäfer, G, Milić, J, Eldahshan, A, Götz, F, Zühlke, K, Schillinger, C, Kreuchwig, A, Elkins, J, Abdul Azeez, K, Oder, A, Moutty, M, Masada, N, Beerbaum, M, Schlegel, B, Niquet, S, Schmieder, P, Krause, G, von Kries, J, Cooper, D, Knapp, S, Rademann, J, Rosenthal, W, Klussmann, E |
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Format: | Journal article |
Language: | English |
Published: |
Wiley
2013
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