Potent achiral agonists of the growth hormone secretagogue (ghrelin) receptor. Part 2: Lead optimisation.

Potent achiral agonists of the growth hormone secretagogue (ghrelin) receptor. Part 2: Lead optimisation.

A series of small molecule orally bioavailable ghrelin receptor agonists have been identified through systematic optimisation of a high throughput screening hit.

Bibliographic Details
Main Authors:	Witherington, J, Abberley, L, Briggs, M, Collis, K, Dean, D, Gaiba, A, King, N, Kraus, H, Shuker, N, Steadman, J, Takle, A, Sanger, G, Wadsworth, G, Butler, S, McKay, F, Muir, A, Winborn, K, Heightman, T
Format:	Journal article
Language:	English
Published:	2008

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