Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

The syntheses and preliminary pharmacological characterisation of two novel cyclic phosphinic acid-containing amino acids designed as conformationally restricted analogues of the metabotropic glutamate receptor agonist AP4 (1) are reported.

Bibliographische Detailangaben
Hauptverfasser:	Conway, S, Miller, J, Bond, A, Clark, B, Jane, D
Format:	Journal article
Sprache:	English
Veröffentlicht:	2002

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