Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4
The syntheses and preliminary pharmacological characterisation of two novel cyclic phosphinic acid-containing amino acids designed as conformationally restricted analogues of the metabotropic glutamate receptor agonist AP4 (1) are reported.
Main Authors: | Conway, S, Miller, J, Bond, A, Clark, B, Jane, D |
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Formato: | Journal article |
Idioma: | English |
Publicado: |
2002
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