Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

The syntheses and preliminary pharmacological characterisation of two novel cyclic phosphinic acid-containing amino acids designed as conformationally restricted analogues of the metabotropic glutamate receptor agonist AP4 (1) are reported.

Номзүйн дэлгэрэнгүй
Үндсэн зохиолчид:	Conway, S, Miller, J, Bond, A, Clark, B, Jane, D
Формат:	Journal article
Хэл сонгох:	English
Хэвлэсэн:	2002

Ижил төстэй зүйлс

Aluminacyclopentanes in the synthesis of 3-substituted phospholanes and α,ω-bisphospholanes
-н: Vladimir A. D’yakonov, зэрэг
Хэвлэсэн: (2016-03-01)

Synthesis of phenylglycine derivatives as potent and selective antagonists of group III metabotropic glutamate receptors.
-н: Conway, S, зэрэг
Хэвлэсэн: (2001)

Metabotropic glutamate receptor agonists for schizophrenia.
-н: Harrison, P
Хэвлэсэн: (2008)

Synthesis of analogues of lycoperdic acid to probe glutamate receptors in the central nervous system
-н: Goundry, W, зэрэг
Хэвлэсэн: (2003)

Synephrine Analogues as Glucocorticoid Receptor Agonists
-н: Eugenia Oleynik, зэрэг
Хэвлэсэн: (2023-11-01)

Structural requirements for selective group III metabotropic glutamate receptor antagonists based on the phenylglycine nucleus.
-н: Jane, D, зэрэг
Хэвлэсэн: (2002)

Novel phenylglycine analogues as potent and selective antagonists of group III mGlu receptors on neonatal rat primary afferent terminals.
-н: Miller, J, зэрэг
Хэвлэсэн: (2000)

Computational study of synthetic agonist ligands of ionotropic glutamate receptors.
-н: Tino Wolter, зэрэг
Хэвлэсэн: (2013-01-01)

Phenylglycine derivatives as antagonists of group III metabotropic glutamate receptors expressed on neonatal rat primary afferent terminals.
-н: Miller, J, зэрэг
Хэвлэсэн: (2003)

The ketamine analogue methoxetamine and 3- and 4-methoxy analogues of phencyclidine are high affinity and selective ligands for the glutamate NMDA receptor.
-н: Bryan L Roth, зэрэг
Хэвлэсэн: (2013-01-01)

Correction: Computational Study of Synthetic Agonist Ligands of Ionotropic Glutamate Receptors
Хэвлэсэн: (2014-01-01)

Correction: Computational Study of Synthetic Agonist Ligands of Ionotropic Glutamate Receptors.
-н: Tino Wolter, зэрэг
Хэвлэсэн: (2014-01-01)

Correction: The Ketamine Analogue Methoxetamine and 3- and 4-Methoxy Analogues of Phencyclidine Are High Affinity and Selective Ligands for the Glutamate NMDA Receptor.
-н: Bryan L Roth, зэрэг
Хэвлэсэн: (2018-01-01)

A new metabotropic glutamate receptor agonist with in vivo anti-allodynic activity
-н: Stanley, N.J., зэрэг
Хэвлэсэн: (2010)

Synthesis of truncated analogues of the iNKT cell agonist, α-galactosyl ceramide (KRN7000), and their biological evaluation
-н: Veerapen, N, зэрэг
Хэвлэсэн: (2011)

Synthesis of truncated analogues of the iNKT cell agonist, α-galactosyl ceramide (KRN7000), and their biological evaluation.
-н: Veerapen, N, зэрэг
Хэвлэсэн: (2011)

Synthesis and Biological Evaluation of Novel Biased Mu-Opioid Receptor Agonists
-н: Yanhao Guo, зэрэг
Хэвлэсэн: (2024-06-01)

Structural insights into neurokinin 3 receptor activation by endogenous and analogue peptide agonists
-н: Wenjing Sun, зэрэг
Хэвлэсэн: (2023-06-01)

Binding site flexibility: Molecular simulation of partial and full agonists within a glutamate receptor
-н: Arinaminpathy, Y, зэрэг
Хэвлэсэн: (2006)

Binding site flexibility: molecular simulation of partial and full agonists within a glutamate receptor.
-н: Arinaminpathy, Y, зэрэг
Хэвлэсэн: (2006)

Effects of glutamate receptor agonists on the P13 auditory evoked potential and startle response in the rat
-н: Christen eSimon, зэрэг
Хэвлэсэн: (2011-01-01)

Direct versatile route to conformationally constrained glutamate analogues
-н: Dyer, J, зэрэг
Хэвлэсэн: (1998)

Group II metabotropic glutamate receptor agonist LY379268 regulates AMPA receptor trafficking in prefrontal cortical neurons.
-н: Min-Juan Wang, зэрэг
Хэвлэсэн: (2013-01-01)

Synthesis and biological evaluation of novel eunicellin analogues
-н: Gilmour, R, зэрэг
Хэвлэсэн: (2005)

Inositol polyphosphates and analogues: synthesis & chemical biology
-н: Shipton, M
Хэвлэсэн: (2021)

The synthesis and biological evaluation of novel eunicellin analogues
-н: Davidson, J, зэрэг
Хэвлэсэн: (2004)

Synthesis and Biological Evaluation of New CRH Analogues
-н: Spyridon Papazacharias, зэрэг
Хэвлэсэн: (2010-01-01)

Synthesis and Biological Evaluation of Aminobisphosphonates—Analogues of Incadronate
-н: Ewa Chmielewska, зэрэг
Хэвлэсэн: (2019-08-01)

Synthesis and Biological Evaluation of Carbocyclic Analogues of Pachastrissamine
-н: Yongseok Kwon, зэрэг
Хэвлэсэн: (2015-02-01)

Molecular determinants of agonist selectivity in glutamate-gated chloride channels which likely explain the agonist selectivity of the vertebrate glycine and GABAA-ρ receptors.
-н: Thomas Blarre, зэрэг
Хэвлэсэн: (2014-01-01)

Minimal Structural Changes Determine Full and Partial Nicotinic Receptor Agonist Activity for Nicotine Analogues
-н: Juan Pablo Gonzalez-Gutierrez, зэрэг
Хэвлэсэн: (2019-07-01)

Defense reaction induced by a metabotropic glutamate receptor agonist microinjected into the dorsal periaqueductal gray of rats
-н: M.L. Molchanov, зэрэг
Хэвлэсэн: (1999-12-01)

The sigma1 receptor agonist enhances long-term depression caused by activation of metabotropic glutamate receptors in rat hippocampal neurons
-н: Pavel D. Rogozin, зэрэг
Хэвлэсэн: (2018-12-01)

Synthesis and Biological Properties of Novel Fluoroprostaglandin Derivatives: Highly Selective and Potent Agonists for Prostaglandin Receptors
-н: Yasushi Matsumuraa, зэрэг
Хэвлэсэн: (2004-03-01)

Correction: Molecular Determinants of Agonist Selectivity in Glutamate-Gated Chloride Channels Which Likely Explain the Agonist Selectivity of the Vertebrate Glycine and GABAA-ρ Receptors
Хэвлэсэн: (2014-01-01)

Correction: Molecular Determinants of Agonist Selectivity in Glutamate-Gated Chloride Channels Which Likely Explain the Agonist Selectivity of the Vertebrate Glycine and GABA-ρ Receptors.
Хэвлэсэн: (2014-01-01)

<it>In vivo </it>antinociception of potent mu opioid agonist tetrapeptide analogues and comparison with a compact opioid agonist - neurokinin 1 receptor antagonist chimera
-н: Guillemyn Karel, зэрэг
Хэвлэсэн: (2012-01-01)

Synthesis of Polyfluorinated KRN7000 Analogues and Biological Implications
-н: M. Isabel Matheu, зэрэг
Хэвлэсэн: (2019-08-01)

Synthesis, reactivity and biological activity of 5-alkoxymethyluracil analogues
-н: Lucie Brulikova, зэрэг
Хэвлэсэн: (2011-05-01)

Glutamate receptor activation is involved in 5-HT2 agonist-induced Arc gene expression in the rat cortex.
-н: Pei, Q, зэрэг
Хэвлэсэн: (2004)