Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

The syntheses and preliminary pharmacological characterisation of two novel cyclic phosphinic acid-containing amino acids designed as conformationally restricted analogues of the metabotropic glutamate receptor agonist AP4 (1) are reported.

Bibliografske podrobnosti
Main Authors:	Conway, S, Miller, J, Bond, A, Clark, B, Jane, D
Format:	Journal article
Jezik:	English
Izdano:	2002

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