Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

The syntheses and preliminary pharmacological characterisation of two novel cyclic phosphinic acid-containing amino acids designed as conformationally restricted analogues of the metabotropic glutamate receptor agonist AP4 (1) are reported.

Sonraí bibleagrafaíochta
Príomhchruthaitheoirí: Conway, S, Miller, J, Bond, A, Clark, B, Jane, D
Formáid: Journal article
Teanga:English
Foilsithe / Cruthaithe: 2002