Re-evaluating the mechanism of action of α,β-unsaturated carbonyl DUB inhibitors B-AP15 and VLX1570: a paradigmatic example of unspecific protein crosslinking with Michael acceptor motif-containing drugs
| Main Authors: | , , , , , , , , , |
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| Format: | Working paper |
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2019
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| _version_ | 1826276333746913280 |
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| author | Ward, J Pinto-Fernandez, A Cornelissen, L Bonham, S Diaz Saez, L Riant, O Huber, K Kessler, B Feron, O Tate, E |
| author_facet | Ward, J Pinto-Fernandez, A Cornelissen, L Bonham, S Diaz Saez, L Riant, O Huber, K Kessler, B Feron, O Tate, E |
| author_sort | Ward, J |
| collection | OXFORD |
| description | |
| first_indexed | 2024-03-06T23:12:23Z |
| format | Working paper |
| id | oxford-uuid:65ecff11-47fb-4010-97c1-19f93fe8ea2b |
| institution | University of Oxford |
| last_indexed | 2024-03-06T23:12:23Z |
| publishDate | 2019 |
| record_format | dspace |
| spelling | oxford-uuid:65ecff11-47fb-4010-97c1-19f93fe8ea2b2022-03-26T18:28:44ZRe-evaluating the mechanism of action of α,β-unsaturated carbonyl DUB inhibitors B-AP15 and VLX1570: a paradigmatic example of unspecific protein crosslinking with Michael acceptor motif-containing drugsWorking paperhttp://purl.org/coar/resource_type/c_8042uuid:65ecff11-47fb-4010-97c1-19f93fe8ea2bSymplectic Elements at Oxford2019Ward, JPinto-Fernandez, ACornelissen, LBonham, SDiaz Saez, LRiant, OHuber, KKessler, BFeron, OTate, E |
| spellingShingle | Ward, J Pinto-Fernandez, A Cornelissen, L Bonham, S Diaz Saez, L Riant, O Huber, K Kessler, B Feron, O Tate, E Re-evaluating the mechanism of action of α,β-unsaturated carbonyl DUB inhibitors B-AP15 and VLX1570: a paradigmatic example of unspecific protein crosslinking with Michael acceptor motif-containing drugs |
| title | Re-evaluating the mechanism of action of α,β-unsaturated carbonyl DUB inhibitors B-AP15 and VLX1570: a paradigmatic example of unspecific protein crosslinking with Michael acceptor motif-containing drugs |
| title_full | Re-evaluating the mechanism of action of α,β-unsaturated carbonyl DUB inhibitors B-AP15 and VLX1570: a paradigmatic example of unspecific protein crosslinking with Michael acceptor motif-containing drugs |
| title_fullStr | Re-evaluating the mechanism of action of α,β-unsaturated carbonyl DUB inhibitors B-AP15 and VLX1570: a paradigmatic example of unspecific protein crosslinking with Michael acceptor motif-containing drugs |
| title_full_unstemmed | Re-evaluating the mechanism of action of α,β-unsaturated carbonyl DUB inhibitors B-AP15 and VLX1570: a paradigmatic example of unspecific protein crosslinking with Michael acceptor motif-containing drugs |
| title_short | Re-evaluating the mechanism of action of α,β-unsaturated carbonyl DUB inhibitors B-AP15 and VLX1570: a paradigmatic example of unspecific protein crosslinking with Michael acceptor motif-containing drugs |
| title_sort | re evaluating the mechanism of action of α β unsaturated carbonyl dub inhibitors b ap15 and vlx1570 a paradigmatic example of unspecific protein crosslinking with michael acceptor motif containing drugs |
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