Extended peptide-based inhibitors efficiently target the proteasome and reveal overlapping specificities of the catalytic beta-subunits.

Eitemau Tebyg

• Solid phase synthesis of peptide vinyl sulfone and peptide epoxyketone proteasome inhibitors
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  Cyhoeddwyd: (2000)
• Activity probe for in vivo profiling of the specificity of proteasome inhibitor bortezomib.
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  Cyhoeddwyd: (2005)
• A cell-permeable inhibitor and activity-based probe for the caspase-like activity of the proteasome.
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  Cyhoeddwyd: (2007)
• Proteasome activity profiling: a simple, robust and versatile method revealing subunit-selective inhibitors and cytoplasmic, defense-induced proteasome activities.
  gan: Gu, C, et al.
  Cyhoeddwyd: (2010)
• Subunit-selective proteasome activity profiling uncovers uncoupled proteasome subunit activities during bacterial infections
  gan: Misas-Villamil, J, et al.
  Cyhoeddwyd: (2017)