A short stereoselective total synthesis of the fusarium toxin equisetin.
A short stereoselective synthesis of the fusarium toxin equisetin, an N-methylserine-derived acyl tetramic acid and potent inhibitor of HIV-1 integrase enzyme, is described using as the key step a stereoselective lithium perchlorate mediated intramolecular Diels-Alder reaction of a fully conjugated...
Hlavní autoři: | , , , |
---|---|
Médium: | Journal article |
Jazyk: | English |
Vydáno: |
2000
|