Developing inhibitors of bromodomain-histone interactions

<p>Lysine acetylation is a widespread protein post-translational modification that influences diverse cellular processes. An association between acetylation of histone N-terminal tails and transcriptional activation has been recognised since the 1960s. However, it has only become apparent sinc...

Descrizione completa

Dettagli Bibliografici
Autore principale: Hewings, D
Altri autori: Conway, S
Natura: Tesi
Lingua:English
Pubblicazione: 2014
Soggetti: