Bicyclic lactams derived from serine or cysteine and 2-methylpropanal

Bicyclic lactams derived from serine or cysteine and 2-methylpropanal

Bicyclic lactams may be prepared from serine or cysteine and 2-methylpropanal; the resulting S,N-heterocycles are more stable than the corresponding O,N-heterocycles but both are synthetic intermediates capable of further elaboration.

Sonraí bibleagrafaíochta
Príomhchruthaitheoirí:	Bagum, H, Shire, BR, Christensen, KE, Genov, M, Pretsch, A, Pretsch, D, Moloney, MG
Formáid:	Journal article
Teanga:	English
Foilsithe / Cruthaithe:	Thieme Publishing 2020

Míreanna comhchosúla

Synthetic access to 3,4-disubstituted pyroglutamates from tetramate derivatives from serine, allo-threonine and cysteine
de réir: Bagum, H, et al.
Foilsithe / Cruthaithe: (2019)

Synthetic access to 3-substituted pyroglutamic acids from tetramate derivatives of serine, threonine, allo-threonine, and cysteine
de réir: Bagum, H, et al.
Foilsithe / Cruthaithe: (2019)

Functionalised bicyclic tetramates derived from cysteine as antibacterial agents.
de réir: Panduwawala, TD, et al.
Foilsithe / Cruthaithe: (2019)

Synthetic access to hydrophilic tetramate derivatives of cysteine
de réir: Zhang, R, et al.
Foilsithe / Cruthaithe: (2020)

Tricyclic Fused Lactams by Mukaiyama Cyclisation of Phthalimides and Evaluation of their Biological Activity
de réir: Lewis T. Ibbotson, et al.
Foilsithe / Cruthaithe: (2022-12-01)

Antibacterial mimics of natural products by side-chain functionalization of bicyclic tetramic acids
de réir: Josa-Cullere, L, et al.
Foilsithe / Cruthaithe: (2018)

Metal binding and its amelioration in tetramates
de réir: Zhang, R, et al.
Foilsithe / Cruthaithe: (2021)

Stereoselective oxygenation of bicyclic lactams
de réir: Cottrell, I, et al.
Foilsithe / Cruthaithe: (2004)

On the diastereoselectivity of alkylations of bicyclic lactams
de réir: Bailey, J, et al.
Foilsithe / Cruthaithe: (2000)

Synthesis and Antibacterial Activity of Bicyclic Lactam-Lactones
de réir: Angelov, P, et al.
Foilsithe / Cruthaithe: (2011)

Prolongation of metallothionein induction combats Aß and α-synuclein toxicity in aged transgenic Caenorhabditis elegans
de réir: Pretsch, D, et al.
Foilsithe / Cruthaithe: (2020)

Enantiopure bicyclic piperidinones: stereoselectivity in lactam enolate alkylations.
de réir: Brewster, A, et al.
Foilsithe / Cruthaithe: (2004)

Uncatalysed diaryldiazo cyclopropanations on bicyclic lactams: access to annulated prolines.
de réir: Harris, L, et al.
Foilsithe / Cruthaithe: (2015)

Non‐Hydrolytic β‐Lactam Antibiotic Fragmentation by l,d‐Transpeptidases and Serine β‐Lactamase Cysteine Variants
de réir: Lohans, C, et al.
Foilsithe / Cruthaithe: (2018)

Propane, butane and 2-Methylpropane/
de réir: International Union of Pure and Applied Chemistry. Analytical Chemistry Division. Commission on Solubility Data, et al.
Foilsithe / Cruthaithe: (1986)

Alkylation of phenylglycinol-derived bicyclic lactams. Enantioselective synthesis of 3-alkylpiperidines
de réir: Mercedes Amat, et al.
Foilsithe / Cruthaithe: (2005-03-01)

Tables of spectral data for structure determination of organic compounds/
de réir: Pretsch, Erno
Foilsithe / Cruthaithe: (1983)

Chemical Sensors and Computer-Aided Analytical Chemistry
de réir: Ernö Pretsch
Foilsithe / Cruthaithe: (1997-10-01)

Chemical Sensors and Computer-Aided Analytical Chemistry
de réir: Ernö Pretsch
Foilsithe / Cruthaithe: (1997-10-01)

2-Methylpropan-2-aminium 4-hydroxybenzoate
de réir: Shu-Lan Yu
Foilsithe / Cruthaithe: (2010-07-01)

SYNTHESIS OF A BICYCLIC GAMMA-LACTAM DIPEPTIDE ANALOG
de réir: Baldwin, J, et al.
Foilsithe / Cruthaithe: (1992)

SYNTHESIS OF A BICYCLIC GAMMA-LACTAM DIPEPTIDE ANALOG
de réir: Baldwin, J, et al.
Foilsithe / Cruthaithe: (1993)

Thionation of bicyclic ß-lactam compounds by Lawesson’s reagent
de réir: Andrés A. Poeylaut Palena, et al.
Foilsithe / Cruthaithe: (2006-01-01)

Synthesis of bicyclic lactams using novel Schmidt reactions
de réir: Mike Casey, et al.
Foilsithe / Cruthaithe: (2003-07-01)

Synthesis of a bicyclic oxo-γ-lactam from a simple caprolactam derivative
de réir: Weck, C, et al.
Foilsithe / Cruthaithe: (2017)

Intramolecular aldol ring closures of cysteine derivatives leading to densely functionalised pyroglutamates
de réir: Almahli, H, et al.
Foilsithe / Cruthaithe: (2019)

2-Methylpropan-2-aminium 2-(methoxycarbonyl)benzoate
de réir: Jian Li
Foilsithe / Cruthaithe: (2011-10-01)

Mechanistic insights into the inhibition of serine proteases by monocyclic lactams.
de réir: Wilmouth, R, et al.
Foilsithe / Cruthaithe: (1999)

An archaeal ADP-dependent serine kinase involved in cysteine biosynthesis and serine metabolism
de réir: Yuki Makino, et al.
Foilsithe / Cruthaithe: (2016-11-01)

Sustainable Synthesis of Novel Arylamide L-Cysteine Methyl Esters Peptidomimetic Derivatives: Inhibitors of Serine and Cysteine-like Proteases
de réir: Aline Silveira Serralbo, et al.
Foilsithe / Cruthaithe: (2020-12-01)

Sustainable Synthesis of Novel Arylamide L-Cysteine Methyl Esters Peptidomimetic Derivatives: Inhibitors of Serine and Cysteine-like Proteases
de réir: Adriana Karla Cardoso Amorim Reis, et al.
Foilsithe / Cruthaithe: (2020-12-01)

SYNTHESIS OF A NOVEL BICYCLIC GAMMA-LACTAM ANALOG OF THE 1-OXAPENAMS
de réir: Baldwin, J, et al.
Foilsithe / Cruthaithe: (1989)

FORMATION OF A NOVEL BICYCLIC GAMMA-LACTAM WITH ISOPENICILLIN-N SYNTHASE
de réir: Baldwin, J, et al.
Foilsithe / Cruthaithe: (1989)

ENZYMATIC-SYNTHESIS OF BICYCLIC GAMMA-LACTAMS USING CLAVAMINIC ACID SYNTHASE
de réir: Baldwin, J, et al.
Foilsithe / Cruthaithe: (1992)

Chemo-enzymatic synthesis of bicyclic gamma-lactams using clavaminic acid synthase
de réir: Baldwin, J, et al.
Foilsithe / Cruthaithe: (1997)

An unexpected bicyclic pyrrolidinedione by rearrangement of the β-lactam ring under basic conditions
de réir: Ramón M. Sánchez, et al.
Foilsithe / Cruthaithe: (2009-06-01)

Asymmetric Synthesis and Antimicrobial Activity of Some New Mono and Bicyclic ÃŽÂ²-Lactams
de réir: A. Taslimi, et al.
Foilsithe / Cruthaithe: (2004-11-01)

(SS,2S,3S)-2-(2-Methylpropan-2-sulfinamido)-3-phenylbutyronitrile
de réir: Klaus Harms, et al.
Foilsithe / Cruthaithe: (2009-11-01)

Bicyclic boronate VNRX-5133 inhibits metallo- and serine-β-lactamases
de réir: Krajnc, A, et al.
Foilsithe / Cruthaithe: (2019)

Wilhelm Simon: 1929–1992
de réir: Erno Pretsch, et al.
Foilsithe / Cruthaithe: (1993-01-01)