Enantioselective synthesis of 4- and 6-azaindolines by a cation-directed cyclization

Enantioselective synthesis of 4- and 6-azaindolines by a cation-directed cyclization

Functionalized 4- and 6-azaindolines are accessible with high levels of enantioselectivity by the cation-directed cyclization of aminopyridine-derived imines via phase-transfer catalysis. The extension of this methodology to diastereoselective cyclizations is also described.

Chi tiết về thư mục
Những tác giả chính:	Smith, M, Lamb, A, Davey, P, Driver, R, Thompson, A
Định dạng:	Journal article
Được phát hành:	American Chemical Society 2016

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