Synthesis and analysis of Leu-enkephalin analogues containing reverse turn peptidomimetics

Synthesis and analysis of Leu-enkephalin analogues containing reverse turn peptidomimetics

The synthesis and 1H n.m.r. analysis of peptidomimetics of Leu-enkephalin containing bicyclic lactams is described.

Bibliographic Details
Main Authors:	Claridge, T, Hulme, C, Kelly, R, Lee, V, Nash, I, Schofield, C
Format:	Journal article
Language:	English
Published:	1996

Similar Items

Metal-Binding Ability of Leu-Enkephalin, Related Glycoconjugates and Peptidomimetics
by: Zsuzsa Majer, et al.
Published: (2015-12-01)

Synthetic Analogue of Leu-Enkephalin Prevents Endothelial Dysfunction in vitro
by: O. A. Grebenchikov, et al.
Published: (2018-05-01)

Synthetic Analogue of Leu-Enkephalin in COVID-19 (a Prospective Clinical Study)
by: M. A. Magomedov, et al.
Published: (2022-08-01)

The influence of non-opiate analogue of leu-enkephalin to the cardiac consequences of intrauterine hypoxia of albino rats
by: Еlena N. Sazonova, et al.
Published: (2019-12-01)

Phosphorus (V) porphyrin diaxially substituted with Leu-enkephalin
by: Gajewski Mariusz, et al.
Published: (2004-09-01)

Synthesis and conformational analysis of cyclic analogues of inverse gamma-turns.
by: Kaewpet, M, et al.
Published: (2008)

Synthesis of novel sulfide-based cyclic peptidomimetic analogues to solonamides
by: José Brango-Vanegas, et al.
Published: (2019-10-01)

The role of amino acid arginine and nitric oxide system in implementing cardioprotective effect of non-opioid analogue of leu-enkephalin in newborn albino rats after intrauterine hypoxia
by: Elena N. Sazonova, et al.
Published: (2020-12-01)

The effects of a met-enkephalin analogue on ACTH, beta-LPH, beta-endorphin and MET-enkephalin in patients with adrenocortical disease.
by: Gaillard, R, et al.
Published: (1981)

The effect of enkephalin analogue on pituitary hormone release in human obesity.
by: Finer, N, et al.
Published: (1987)

[D-Ala2, D-Leu5] Enkephalin Attenuates Hepatic Ischemia–Reperfusion Injury in Cirrhotic Rats
by: Jueying Liu, et al.
Published: (2022-05-01)

The effects of d-ala2, d-leu5-enkephalin (dadle)"s continuous perfusion on erythrogram and biochemical profile in rats
by: AKYAZI I, et al.
Published: (2013-07-01)

Reversible acylation of elastase by gamma-lactam analogues of beta-lactam inhibitors
by: Westwood, N, et al.
Published: (1997)

The influence of experimental inflammation and axotomy on leucine enkephalin (leuENK) distribution in intramural nervous structures of the porcine descending colon
by: Slawomir Gonkowski, et al.
Published: (2018-05-01)

The behavioural effects of enkephalin analogues injected into the ventral tegmental area and globus pallidus.
by: Joyce, E, et al.
Published: (1981)

Development of peptidomimetic ligands of Pro-Leu-Gly-NH2 as allosteric modulators of the dopamine D2 receptor
by: Swapna Bhagwanth, et al.
Published: (2013-01-01)

An analogue of met-enkephalin attenuates the pituitary-adrenal response to ovine corticotrophin releasing factor.
by: Grossman, A, et al.
Published: (1986)

The opioid control of LH and FSH release: effects of a met-enkephalin analogue and naloxone.
by: Grossman, A, et al.
Published: (1981)

Comments on the use of a dichromophoric circular dichroism assay for the identification of beta-turns in peptides.
by: Baldwin, J, et al.
Published: (1994)

SYNTHESIS OF POTENTIAL BETA-TURN BICYCLIC DIPEPTIDE MIMETICS
by: Baldwin, J, et al.
Published: (1993)

Synthesis, antiproliferative and antimicrobial activities of (KLAKLAK)2-NH2 analogue containing nor-Leu and its conjugates with a second pharmacophore
by: Sirine Jaber, et al.
Published: (2023-12-01)

Synthesis and Structural Study of a New β-Turn Inducer Peptidomimetic Incorporating 1-Amino-1-Aminomethylcyclohexane
by: María Campos, et al.
Published: (2021-11-01)

Novel peptidomimetic structures: enantioselective synthesis of conformationally constrained lysine, ornithine and alanine analogues from pyroglutamic acid
by: Goswami, R, et al.
Published: (1999)

Heterocycles in Peptidomimetics and Pseudopeptides: Design and Synthesis
by: Ambra Guarnaccio, et al.
Published: (2012-03-01)

CIRCULATING CATECHOLAMINES, MELATONIN AND ENKEPHALIN IN MAN FOLLOWING ADMINISTRATION OF A MET-ENKEPHALIN ANALOG
by: Grossman, A, et al.
Published: (1982)

Synthesis of novel phosphorylated peptidomimetics which contain ω-haloalkyl and ω-thiocyanoethyl residues
by: Oleksandr V. Golovchenko, et al.
Published: (2020-01-01)

[D-Ala2, D-Leu5]-enkephalin (DADLE) provides protection against myocardial ischemia reperfusion injury by inhibiting Wnt/β-Catenin pathway
by: Linwen Liu, et al.
Published: (2024-02-01)

STUDIES OF ACUTE TOXICITY OF OXAZOLE CONTAINING PEPTIDOMIMETICS AT INTRAGASTRIC ADMINISTRATION
by: K.V. Sedko, et al.
Published: (2016-04-01)

Opiate receptors: enkephalins and endorphins.
by: Grossman, A, et al.
Published: (1983)

An unsaturated peptidomimetic assembly derived from a carbohydrate.
by: Chung, Y, et al.
Published: (2004)

An Effective and Safe Enkephalin Analog for Antinociception
by: K. K. DurgaRao Viswanadham, et al.
Published: (2021-06-01)

Developmental-Based Classification of Enkephalin and Somatostatin Containing Neurons of the Chicken Central Extended Amygdala
by: Alessandra Pross, et al.
Published: (2022-05-01)

The Involvement of Endogenous Enkephalins in Glucose Homeostasis
by: Vanessa Escolero, et al.
Published: (2023-02-01)

Delta opioid peptide [d-Ala2, d-Leu5] enkephalin confers neuroprotection by activating delta opioid receptor-AMPK-autophagy axis against global ischemia
by: Zelin Lai, et al.
Published: (2020-06-01)

Delta Opioid Peptide [d-Ala2, d-Leu5] Enkephalin (DADLE) Exerts a Cytoprotective Effect in Astrocytes Exposed to Oxygen-Glucose Deprivation by Inducing Autophagy
by: Shuyan Wang, et al.
Published: (2019-06-01)

FRAGMENTATION OF RGD-PEPTIDOMIMETICS CONTAINING PIPERAZINE FRAGMENT IN FAB MASS SPECTROMETRY CONDITIONS
by: A. I. Gren, et al.
Published: (2016-04-01)

Synthesis of imidazo[1,2-a]pyridine-containing peptidomimetics by tandem of Groebke–Blackburn–Bienaymé and Ugi reactions
by: Oleksandr V. Kolomiiets, et al.
Published: (2023-05-01)

Asymmetric synthesis of propargylamines as amino acid surrogates in peptidomimetics
by: Matthias Wünsch, et al.
Published: (2017-11-01)

Conformational Preferences and Antiproliferative Activity of Peptidomimetics Containing Methyl 1′-Aminoferrocene-1-carboxylate and Turn-Forming Homo- and Heterochiral Pro-Ala Motifs
by: Monika Kovačević, et al.
Published: (2021-12-01)

Synthetic leu-enkefalin analogue prevents activation of neutrophils induced by a bacterial component
by: O. A. Grebenchikov, et al.
Published: (2019-07-01)