Novel 2-oxoglutarate analogues modulate the epigenetic activity of the cancer-related human enzyme aspartate/asparagine-β-hydroxylase

Geahča maid

• Synthesis of 2-oxoglutarate derivatives and their evaluation as cosubstrates and inhibitors of human aspartate/asparagine-β-hydroxylase
  Dahkki: Brewitz, L, et al.
  Almmustuhtton: (2020)
• Kinetic parameters of human aspartate/asparagine-β-hydroxylase suggest that it has a possible function in oxygen sensing
  Dahkki: Brewitz, L, et al.
  Almmustuhtton: (2020)
• Synthesis of novel pyridine-carboxylates as small-molecule inhibitors of human aspartate/asparagine-β-hydroxylase
  Dahkki: Brewitz, L, et al.
  Almmustuhtton: (2020)
• Aspartate/asparagine-β-hydroxylase: a high-throughput mass spectrometric assay for discovery of small molecule inhibitors
  Dahkki: Brewitz, L, et al.
  Almmustuhtton: (2020)
• Aspartate/asparagine-β-hydroxylase: a high-throughput mass spectrometric assay for discovery of small molecule inhibitors
  Dahkki: Lennart Brewitz, et al.
  Almmustuhtton: (2020-05-01)