Tandem copper-catalysed aryl and alkenyl amination reactions: the synthesis of N-functionalised indoles.
A Cu-diamine complex effectively catalyses tandem C-N bond formation on 2-(2-haloalkenyl)-aryl halide substrates, to deliver a series of N-functionalised indoles. Anilines, amides and carbamates are all effective coupling partners under the developed conditions.
Hauptverfasser: | , , |
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Format: | Journal article |
Sprache: | English |
Veröffentlicht: |
2009
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Zusammenfassung: | A Cu-diamine complex effectively catalyses tandem C-N bond formation on 2-(2-haloalkenyl)-aryl halide substrates, to deliver a series of N-functionalised indoles. Anilines, amides and carbamates are all effective coupling partners under the developed conditions. |
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