Tandem copper-catalysed aryl and alkenyl amination reactions: the synthesis of N-functionalised indoles.
A Cu-diamine complex effectively catalyses tandem C-N bond formation on 2-(2-haloalkenyl)-aryl halide substrates, to deliver a series of N-functionalised indoles. Anilines, amides and carbamates are all effective coupling partners under the developed conditions.
| Główni autorzy: | , , |
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| Format: | Journal article |
| Język: | English |
| Wydane: |
2009
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| Streszczenie: | A Cu-diamine complex effectively catalyses tandem C-N bond formation on 2-(2-haloalkenyl)-aryl halide substrates, to deliver a series of N-functionalised indoles. Anilines, amides and carbamates are all effective coupling partners under the developed conditions. |
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