Diastereoselective synthesis of pyrrolidine derivatives via a one-pot nitro-Mannich/hydroamination cascade using base and gold catalysis.

Diastereoselective synthesis of pyrrolidine derivatives via a one-pot nitro-Mannich/hydroamination cascade using base and gold catalysis.

An efficient one-pot nitro-Mannich/hydroamination cascade reaction for the synthesis of substituted pyrrolidines bearing three stereocentres is reported. Proceeding under the control of a combination of base and gold(I) catalysts, the cascade reaction affords the pyrrolidine products in high yields...

पूर्ण विवरण

ग्रंथसूची विवरण
मुख्य लेखकों:	Ďuriš, A, Barber, D, Sanganee, H, Dixon, D
स्वरूप:	Journal article
भाषा:	English
प्रकाशित:	2013

समान संसाधन

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