Azasugar analogues: conformationally restricted vicinal diamine derived from (S)-(-)-pyroglutamic acid

Azasugar analogues: conformationally restricted vicinal diamine derived from (S)-(-)-pyroglutamic acid

The preparation of a diamino substituted pyrrolidinone system in a diastereoselectively controlled manner is described. The procedure employed made use of electrophilic amination of a chiral bicyclic γ-lactam, which when subjected to sequential deprotection provided a simple route to a 3,4- diaminop...

書目詳細資料
Main Authors:	Chan, P, Cottrell, I, Moloney, M
格式:	Journal article
語言:	English
出版:	1999

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