Azasugar analogues: conformationally restricted vicinal diamine derived from (S)-(-)-pyroglutamic acid

Azasugar analogues: conformationally restricted vicinal diamine derived from (S)-(-)-pyroglutamic acid

The preparation of a diamino substituted pyrrolidinone system in a diastereoselectively controlled manner is described. The procedure employed made use of electrophilic amination of a chiral bicyclic γ-lactam, which when subjected to sequential deprotection provided a simple route to a 3,4- diaminop...

Cur síos iomlán

Sonraí bibleagrafaíochta
Príomhchruthaitheoirí:	Chan, P, Cottrell, I, Moloney, M
Formáid:	Journal article
Teanga:	English
Foilsithe / Cruthaithe:	1999

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