Design of a chemical probe for the bromodomain and plant homeodomain finger-containing (BRPF) family of proteins
The bromodomain and plant homeodomain finger-containing (BRPF) family are scaffolding proteins important for the recruitment of histone acetyltransferases of the MYST family to chromatin. Here, we describe NI-57 (16) as new pan-BRPF chemical probe of the bromodomain (BRD) of the BRPFs. Inhibitor 16...
Autors principals: | , , , , , , , , , , , , , , , , |
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Format: | Journal article |
Idioma: | English |
Publicat: |
American Chemical Society
2017
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