Palladium catalysed elaboration of codeine and morphine

Palladium catalysed elaboration of codeine and morphine

Palladium catalysed coupling reactions of 6-O-tert-butyldimethylsilyl-1-bromocodeine and 6-O-tert-butyldimethylsilyl-3-trifluoromethylsulfonylmorphine allow a range of substituted analogues of codeine in the 1-position and morphine in the 3-position to be efficiently and selectively prepared.

Dades bibliogràfiques
Autors principals:	Davies, S, Goodwin, C, Pyatt, D, Smith, A
Format:	Journal article
Idioma:	English
Publicat:	2001

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