Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety

Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety

Hiển thị phiên bản (1) khác

A series of 3-methylidene-1H-indol-2(3H)-ones substituted with a 5- or 6-pentafluorosulfanyl group has been synthesized by a Knoevenagel condensation reaction of SF5-substituted oxindoles with a range of aldehydes. The resulting products were characterized by X-ray crystallography studies and were t...

Mô tả đầy đủ

Chi tiết về thư mục
Những tác giả chính:	Sansook, S, Ocasio, CA, Day, IJ, Tizzard, GJ, Coles, SJ, Fedorov, O, Bennett, JM, Elkins, JM, Spencer, J
Định dạng:	Journal article
Ngôn ngữ:	English
Được phát hành:	Royal Society of Chemistry 2017

Những quyển sách tương tự

Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety
Bằng: Sansook, S, et al.
Được phát hành: (2017)

Synthesis of Aryl Propionamide Scaffold Containing a Pentafluorosulfanyl Moiety as SARMs
Bằng: Pingxuan Shao, et al.
Được phát hành: (2019-11-01)

Expanding the repertoire of low-molecular-weight pentafluorosulfanyl-substituted scaffolds
Bằng: Jose, A, et al.
Được phát hành: (2022)

Targeting the water network in cyclin G-associated kinase (GAK) with 4-anilino-quin(az)oline inhibitors
Bằng: Asquith, CRM, et al.
Được phát hành: (2020)

Pentafluorosulfanyl-containing Triclocarban Analogs with Potent Antimicrobial Activity
Bằng: Eugènia Pujol, et al.
Được phát hành: (2018-11-01)

Novel pentafluorosulfanyl-containing triclocarban analogs selectively kill Gram-positive bacteria
Bằng: Ali Pormohammad, et al.
Được phát hành: (2024-06-01)

Recent achievements in the synthesis and reactivity of pentafluorosulfanyl-alkynes
Bằng: René, Floriane, et al.
Được phát hành: (2024-11-01)

Probing the Anticancer Action of Novel Ferrocene Analogues of MNK Inhibitors
Bằng: Supojjanee Sansook, et al.
Được phát hành: (2018-08-01)

Synthesis and Properties of Pentafluorosulfanyl Group (SF<sub>5</sub>)-Containing Meta-Diamide Insecticides
Bằng: Jae Gon Kim, et al.
Được phát hành: (2020-11-01)

Modular synthesis of di- and trisubstituted imidazoles from ketones and aldehydes: a route to kinase inhibitors
Bằng: De Toledo, I, et al.
Được phát hành: (2019)

Identification of a New Pentafluorosulfanyl-Substituted Chalcone with Activity Against Hepatoma and Human Parasites
Bằng: Alessandra Viperino, et al.
Được phát hành: (2025-01-01)

Synthesis and nucleophilic aromatic substitution of 3-fluoro-5-nitro-1-(pentafluorosulfanyl)benzene
Bằng: Javier Ajenjo, et al.
Được phát hành: (2016-02-01)

Identification and optimization of 4-anilinoquinolines as inhibitors of cyclin G associated kinase
Bằng: Asquith, C, et al.
Được phát hành: (2017)

Research Progress in HIV and Mycobacterium tuberculosis Inhibitors Containing Sulfonamide Moiety
Bằng: Christiana Abimbola Salubi
Được phát hành: (2023-01-01)

Using the negative hyperconjugation effect of pentafluorosulfanyl acceptors to enhance two-photon absorption in push–pull chromophores
Bằng: Gautam, Prabhat, et al.
Được phát hành: (2020)

Exploring kinase family inhibitors and their moiety preferences using deep SHapley additive exPlanations
Bằng: You-Wei Fan, et al.
Được phát hành: (2022-06-01)

Development of Hydroxamate Derivatives Containing a Pyrazoline Moiety as APN Inhibitors to Overcome Angiogenesis
Bằng: Yangyang Liu, et al.
Được phát hành: (2022-11-01)

Synthesis of new 1, 8-dioxo-octahydroxanthene derivatives containing 4-thiazolidinone moiety containing 4-thiazolidinone moiety
Bằng: Maryam Robati, et al.
Được phát hành: (2017-10-01)

Synthesis of Pyridinium Moiety Containing Triazolyl Purines
Bằng: Aleksejs Burcevs, et al.
Được phát hành: (2024-07-01)

Design and analysis of the 4-anilino-quin(az)oline kinase inhibition profiles of GAK/SLK/STK10 using quantitative structure activity relationships
Bằng: Asquith, C, et al.
Được phát hành: (2019)

Identification of pan-kinase-family inhibitors using graph convolutional networks to reveal family-sensitive pre-moieties
Bằng: Xiang-Yu Lin, et al.
Được phát hành: (2022-06-01)

Chemical probes for understudied kinases: challenges and opportunities
Bằng: Serafim, RAM, et al.
Được phát hành: (2021)

Novel amide derivatives containing azetidine moiety as potential SDH inhibitors: Design, synthesis, and evaluation of bioactivity
Bằng: Yong Zhang, et al.
Được phát hành: (2024-05-01)

Binding and structural analyses of potent inhibitors of the human Ca2+/calmodulin dependent protein kinase kinase 2 (CAMKK2) identified from a collection of commercially-available kinase inhibitors.
Bằng: Profeta, GS, et al.
Được phát hành: (2019)

Studies of Halogen Bonding Induced by Pentafluorosulfanyl Aryl Iodides: A Potential Group of Halogen Bond Donors in a Rational Drug Design
Bằng: Yuji Sumii, et al.
Được phát hành: (2019-10-01)

Synthesis and Characterization of Some Compounds containing Pyrazole Moiety
Bằng: Samer M. Tayib, et al.
Được phát hành: (2018-11-01)

Synthesis of Crown Ethers Containing a Rubicene Moiety
Bằng: Mario Smet, et al.
Được phát hành: (2000-03-01)

Synthesis of Some Heterocyclic Compounds Containing Tetrahydroisoquinoline Moiety
Bằng: Mohammad Al-Iraqi, et al.
Được phát hành: (2013-12-01)

Design, Synthesis, and Biological Evaluation of Pyridazinones Containing the (2-Fluorophenyl) Piperazine Moiety as Selective MAO-B Inhibitors
Bằng: Muhammed Çeçen, et al.
Được phát hành: (2020-11-01)

Novel 2-indolinones containing a sulfonamide moiety as selective inhibitors of candida β-carbonic anhydrase enzyme
Bằng: Atilla Akdemir, et al.
Được phát hành: (2019-01-01)

Synthesis and structure-activity relationships of 3,5-disubstituted-pyrrolo[2,3-b]pyridines as inhibitors of adaptor-sssociated kinase 1 with antiviral activity
Bằng: Verdonck, S, et al.
Được phát hành: (2019)

Synthesis of chloro-substituted liquid crystal containing Azobenzene moieties
Bằng: Sylvester Julius
Được phát hành: (2008)

Synthesis and Fungicidal Activity of Pyrazolecarboxamide Containing α-Aminoacetanilide Moiety
Bằng: Zhi-Yong Fang, et al.
Được phát hành: (2012-01-01)

Biginelli Synthesis of Novel Dihydropyrimidinone Derivatives Containing Phthalimide Moiety
Bằng: Mashooq A. Bhat, et al.
Được phát hành: (2020-01-01)

Spiropyrans Containing the Reactive Substituents in the 2H-Chromene Moiety
Bằng: B. S. Lukyanov, et al.
Được phát hành: (2007-01-01)

Antioxidant and anticancer activities of α-aminophosphonates containing thiadiazole moiety
Bằng: Mohamed M. Azaam, et al.
Được phát hành: (2018-01-01)

Synthesis and Antiviral Bioactivities of ÃŽÂ±-Aminophosphonates Containing Alkoxyethyl Moieties
Bằng: Zhuo Chen, et al.
Được phát hành: (2006-09-01)

Synthesis of some new hydrazone derivatives containing benzothiazole moiety
Bằng: Özdemir Ahmet, et al.
Được phát hành: (2012-01-01)

Antidepressant potential of nitrogen-containing heterocyclic moieties: An updated review
Bằng: Nadeem Siddiqui, et al.
Được phát hành: (2011-01-01)

The spectrogram data of quinazoline derivatives containing a dithioacetal moiety
Bằng: Dandan Xie, et al.
Được phát hành: (2018-10-01)