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1
Arylsulfonyl fluoride boronic acids: preparation and coupling reactivity
Published 2019“…The boronic acids undergo efficient Sukuki-Miyaura coupling reactions with a range of aryl halides. …”
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2
Boronic acid catalyzed ene carbocyclization of acetylenic dicarbonyl compounds.
Published 2010Journal article -
3
B-11 NMR-STUDIES OF AN ARYL BORONIC ACID BOUND TO CHYMOTRYPSIN AND SUBTILISIN
Published 1991“…The binding of aryl boronic acids to α-chymotrypsin and subtilisin has been studied by 11B NMR spectroscopy; evidence is provided for the direct spectroscopic observation of a tetrahedral enzyme/boromate complex. © 1991.…”
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4
Highly enantioselective rhodium-catalyzed cross-coupling of boronic acids and racemic allyl halides
Published 2019“…The method couples racemic allyl halide starting materials with sp2-hybridized boronic acid derivatives and is compatible with heterocyclic coupling partners. …”
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5
Single-molecule determination of the isomers of D-glucose and D-fructose that bind to boronic acids
Published 2018“…Monosaccharides, such as D-glucose and D-fructose, exist in aqueous solution as an equilibrium mixture of cyclic isomers and can be detected with boronic acids by the reversible formation of boronate esters. …”
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6
Dynamic combinatorial chemistry employing boronic acids/boronate esters leads to potent oxygenase inhibitors.
Published 2012“…Dynamic duo: The reversible reaction of boronic acids with alcohols to form boronate esters, coupled to protein mass spectrometry analyses, was used to discover potent oxygenase inhibitors. …”
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7
A boronic-acid-based probe for fluorescence polarization assays with penicillin binding proteins and β-lactamases
Published 2011Journal article -
8
A boronic-acid-based probe for fluorescence polarization assays with penicillin binding proteins and β-lactamases.
Published 2012“…We report the development of a fluorescence polarization (FP) assay for PBPs and "serine" β-lactamases using a boronic-acid-based, reversibly binding "tracer." The tracer was designed based on a crystal structure of a covalent complex between a boronic acid and PBP1b from Streptococcus pneumoniae. …”
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9
Synthesis of 18F-difluoromethylarenes using aryl boronic acids, ethyl bromofluoroacetate and [18F]fluoride
Published 2019Journal article -
10
DIRECT OBSERVATION OF A TETRAHEDRAL BORONIC ACID BETA-LACTAMASE COMPLEX USING B-11 NMR-SPECTROSCOPY
Published 1991“…A tetrahedral boronic acid-β-lactamase complex formed by treatment of the P99 β-lactamase enzyme from Enterobacter cloacae with 3-dansylamidophenylboronic acid has been directly observed using 11B NMR spectroscopy.…”
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11
Nickel(II)-catalyzed synthesis of sulfinates from aryl and heteroaryl boronic acids and the sulfur dioxide surrogate DABSO
Published 2019Journal article -
12
Carbon-carbon bond construction using boronic acids and aryl methyl sulfides: orthogonal reactivity in Suzuki-type couplings
Published 2013“…The Rh(i)-catalysed coupling of aryl and alkenyl boronic acids with simple aryl and alkenyl methyl sulfides is reported. …”
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13
Palladium(II)-catalyzed synthesis of sulfinates from boronic acids and DABSO: a redox-neutral, phosphine-free transformation
Published 2016“…A redox-neutral palladium(II)-catalyzed conversion of aryl, heteroaryl, and alkenyl boronic acids into sulfinate intermediates, and onwards to sulfones and sulfonamides, has been realized. …”
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14
Radiosynthesis of [18F]ArylSCF2H using aryl boronic acids, S-(chlorofluoromethyl)benzenesulfonothioate and [18F]fluoride
Published 2020“…Herein, we report a mild and practical protocol for the copper-catalyzed chlorofluoromethylthiolation of (hetero)aryl boronic acids with the novel reagent PhSO2SCFClH. The resulting products are amenable to halogen exchange 18F-fluorination with cyclotron-produced [18F]fluoride affording [18F]ArSCF2H. …”
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15
Sequential catalysis: Exploiting a single rhodium(I) catalyst to promote an alkyne hydroacylation–aryl boronic acid conjugate addition sequence
Published 2016“…We demonstrate that a single Rh(I) complex can promote two mechanistically distinct C-C bond-forming reactions – alkyne hydroacylation and aryl boronic acid conjugate addition – to deliver substituted ketone products from the controlled assembly of three readily available fragments. …”
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16
Enantioselective three-component assembly of β’-aryl-enones using a rhodium-catalyzed alkyne hydroacylation/aryl boronic acid conjugate addition sequence
Published 2017“…The sequence corresponds to the formal regio- and enantioselective mono-conjugate addition of aryl boronic acids to dienones.…”
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17
Synthesis and evaluation of 3-(dihydroxyboryl)benzoic acids as D,D-carboxypeptidase R39 inhibitors.
Published 2009“…Here we report aromatic boronic acid inhibitors of the D,D-carboxypeptidase R39 from Actinomadura sp. strain. …”
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18
Arylations mediated by lead(IV) in the presence of formazan and imine ligands
Published 2009“…The use of formazan and imine ligands in arylations of β-dicarbonyl systems by phenyl boronic acid/lead(IV) carboxylates is examined. © 2009 Elsevier Ltd. …”
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19
Structure guided development of potent reversibly binding penicillin binding protein inhibitors.
Published 2011“…Following from the evaluation of different types of electrophiles, combined modeling and crystallographic analyses are used to generate potent boronic acid based inhibitors of a penicillin binding protein. …”
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20
Spatially resolved Suzuki coupling reaction initiated and controlled using a catalytic AFM probe.
Published 2005“…Herein we report a chemically specific Suzuki coupling reaction between a surface-confined aryl bromide and boronic acid reagents in solution achieved using a catalytic AFM probe.…”
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