Development and application of in silico models to design new antibacterial 5-amino-4-cyano-1,3-oxazoles against colistin-resistant E. coli strains by Ivan Semenyuta, Diana Hodyna, Vasyl Kovalishyn, Bohdan Demydchuk, Maryna Kachaeva, Stepan Pilyo, Volodymyr Brovarets, Larysa Metelytsia

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Delta Sleep-Inducing Peptide Recovers Motor Function in SD Rats after Focal Stroke by Elena A. Tukhovskaya, Alina M. Ismailova, Elvira R. Shaykhutdinova, Gulsara A. Slashcheva, Igor A. Prudchenko, Inessa I. Mikhaleva, Oksana N. Khokhlova, Arkady N. Murashev, Vadim T. Ivanov

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Sea Anemone Kunitz-Type Peptides Demonstrate Neuroprotective Activity in the 6-Hydroxydopamine Induced Neurotoxicity Model by Oksana Sintsova, Irina Gladkikh, Margarita Monastyrnaya, Valentin Tabakmakher, Ekaterina Yurchenko, Ekaterina Menchinskaya, Evgeny Pislyagin, Yaroslav Andreev, Sergey Kozlov, Steve Peigneur, Jan Tytgat, Dmitry Aminin, Emma Kozlovskaya, Elena Leychenko

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Alkyl Derivatives of Perylene Photosensitizing Antivirals: Towards Understanding the Influence of Lipophilicity by Igor E. Mikhnovets, Jiří Holoubek, Irina S. Panina, Jan Kotouček, Daniil A. Gvozdev, Stepan P. Chumakov, Maxim S. Krasilnikov, Mikhail Y. Zhitlov, Evgeny L. Gulyak, Alexey A. Chistov, Timofei D. Nikitin, Vladimir A. Korshun, Roman G. Efremov, Vera A. Alferova, Daniel Růžek, Luděk Eyer, Alexey V. Ustinov

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Recombinant Analogs of Sea Anemone Kunitz-Type Peptides Influence P2X7 Receptor Activity in Neuro-2a Cells by Evgeny A. Pislyagin, Ekaterina S. Menchinskaya, Irina N. Gladkikh, Aleksandra N. Kvetkina, Oksana V. Sintsova, Darya V. Popkova, Sergei A. Kozlovskiy, Tatiana Y. Gorpenchenko, Galina N. Likhatskaya, Leonid A. Kaluzhskiy, Alexis S. Ivanov, Yaroslav A. Andreev, Sergey A. Kozlov, Pavel S. Dmitrenok, Dmitry L. Aminin, Elena V. Leychenko

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1,3-Oxazol-4-ylphosphonium salts as new non-peptide inhibitors of furin by T. V. Osadchuk, V. K. Kibirev1,2, O. V. Shybyryn, A. V. Semyroz, Ye. S. Velihina, Е. R. Abdurakhmanova, V. S. Brovarets

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Combining mKate2-Kv1.3 Channel and Atto488-Hongotoxin for the Studies of Peptide Pore Blockers on Living Eukaryotic Cells by Nikita A. Orlov, Anastasia A. Ignatova, Elena V. Kryukova, Sergey A. Yakimov, Mikhail P. Kirpichnikov, Oksana V. Nekrasova, Alexey V. Feofanov

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Facade-Based Bicelles as a New Tool for Production of Active Membrane Proteins in a Cell-Free System by Marina V. Goncharuk, Ekaterina V. Vasileva, Egor A. Ananiev, Andrey Y. Gorokhovatsky, Eduard V. Bocharov, Konstantin S. Mineev, Sergey A. Goncharuk

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Clenbuterol exerts antidiabetic activity through metabolic reprogramming of skeletal muscle cells by Jaroslawna Meister, Derek B. J. Bone, Jonas R. Knudsen, Luiz F. Barella, Thomas J. Velenosi, Dmitry Akhmedov, Regina J. Lee, Amanda H. Cohen, Oksana Gavrilova, Yinghong Cui, Gerard Karsenty, Min Chen, Lee S. Weinstein, Maximilian Kleinert, Rebecca Berdeaux, Thomas E. Jensen, Erik A. Richter, Jürgen Wess

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Spatial Structure of NanoFAST in the Apo State and in Complex with its Fluorogen HBR-DOM2 by Vladislav A. Lushpa, Nadezhda S. Baleeva, Sergey A. Goncharuk, Marina V. Goncharuk, Alexander S. Arseniev, Mikhail S. Baranov, Konstantin S. Mineev

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Activity Dependence of a Novel Lectin Family on Structure and Carbohydrate-Binding Properties by Irina Chikalovets, Alina Filshtein, Valentina Molchanova, Tatyana Mizgina, Pavel Lukyanov, Olga Nedashkovskaya, Kuo-Feng Hua, Oleg Chernikov

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Exhaustive Search of the Receptor Ligands by the CyCLOPS (Cytometry Cell-Labeling Operable Phage Screening) Technique by Irina A. Ishina, Ioanna N. Filimonova, Maria Y. Zakharova, Leyla A. Ovchinnikova, Azad E. Mamedov, Yakov A. Lomakin, Alexey A. Belogurov

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The Brassica napus L. plants expressing antimicrobial peptide cecropin P1 are safe for colonization by beneficial associative microorganisms by Natalia S. Zakharchenko, Olga V. Furs, Elena B. Rukavtsova, Sergey V. Tarlachkov, Anatolii A. Kosobryukhov, Vladimir D. Kreslavski, Olga V. Dyachenko, Yaroslav I. Buryanov, Taras V. Shevchuk

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Adipocyte β-arrestin-2 is essential for maintaining whole body glucose and energy homeostasis by Sai P. Pydi, Shanu Jain, Wesley Tung, Yinghong Cui, Lu Zhu, Wataru Sakamoto, Shalini Jain, Brent S. Abel, Monica C. Skarulis, Jie Liu, Thanh Huynh, Karel Pacak, Marc G. Caron, Oksana Gavrilova, Toren Finkel, Jürgen Wess

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Stereochemical course of hydrolytic reaction catalyzed by alpha-galactosidase from cold adaptable marine bacterium of genus Pseudoalteromonas by Irina Yu Bakunina, Larissa A Balabanova, Vasiliy A Golotin, Lyubov V Slepchenko, Lyubov V Slepchenko, Vladimir V Isakov, Valeriy A Rasskazov

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Membrane-Disrupting Activity of Cobra Cytotoxins Is Determined by Configuration of the N-Terminal Loop by Peter V. Dubovskii, Anastasia A. Ignatova, Anna S. Alekseeva, Vladislav G. Starkov, Ivan A. Boldyrev, Alexey V. Feofanov, Yuri N. Utkin

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Cytotoxic Drimane-Type Sesquiterpenes from Co-Culture of the Marine-Derived Fungi <i>Aspergillus carneus</i> KMM 4638 and <i>Beauveria felina</i> (=<i>Isaria felina</i>) KMM 4639 by Olesya I. Zhuravleva, Elena B. Belousova, Galina K. Oleinikova, Alexandr S. Antonov, Yuliya V. Khudyakova, Anton B. Rasin, Roman S. Popov, Ekaterina S. Menchinskaya, Phan Thi Hoai Trinh, Anton N. Yurchenko, Ekaterina A. Yurchenko

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Zosteropenillines: Polyketides from the MarineDerived Fungus Penicillium thomii by Shamil Sh. Afiyatullov, Elena V. Leshchenko, Dmitrii V. Berdyshev, Maria P. Sobolevskaya, Alexandr S. Antonov, Vladimir A. Denisenko, Roman S. Popov, Mikhail V. Pivkin, Anatoly A. Udovenko, Evgeny A. Pislyagin, Gunhild von Amsberg, Sergey A. Dyshlovoy

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Amphiphilic Poly(<i>N</i>-vinylpyrrolidone) Nanoparticles Conjugated with DR5-Specific Antitumor Cytokine DR5-B for Targeted Delivery to Cancer Cells by Anne Yagolovich, Andrey Kuskov, Pavel Kulikov, Leily Kurbanova, Dmitry Bagrov, Artem Artykov, Marine Gasparian, Svetlana Sizova, Vladimir Oleinikov, Anastasia Gileva, Mikhail Kirpichnikov, Dmitry Dolgikh, Elena Markvicheva

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New Three-Finger Protein from Starfish <i>Asteria rubens</i> Shares Structure and Pharmacology with Human Brain Neuromodulator Lynx2 by Alexander S. Paramonov, Mikhail A. Shulepko, Alexey M. Makhonin, Maxim L. Bychkov, Dmitrii S. Kulbatskii, Andrey M. Chernikov, Mikhail Yu. Myshkin, Sergey V. Shabelnikov, Zakhar O. Shenkarev, Mikhail P. Kirpichnikov, Ekaterina N. Lyukmanova

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