A Web Server for GPCR-GPCR Interaction Pair Prediction by Wataru Nemoto, Wataru Nemoto, Yoshihiro Yamanishi, Vachiranee Limviphuvadh, Shunsuke Fujishiro, Sakie Shimamura, Aoi Fukushima, Hiroyuki Toh

Subjects: “…GPCR…”
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Corrigendum: A Web Server for GPCR-GPCR Interaction Pair Prediction by Wataru Nemoto, Wataru Nemoto, Yoshihiro Yamanishi, Vachiranee Limviphuvadh, Shunsuke Fujishiro, Sakie Shimamura, Aoi Fukushima, Hiroyuki Toh

Subjects: “…GPCR…”
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Holistic concepts in GPCR dynamics by Kota Katayama, Ryoji Suno

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Discovery of Pathologic GPCR Aggregation by Ursula Quitterer, Ursula Quitterer, Said AbdAlla

“…Mechanisms underlying GPCR activation and signaling are therefore of great pharmacologic interest. …”
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GPCR oligomers in pharmacology and signaling by González-Maeso Javier

“…When activated by an agonist, the GPCR undergoes conformational changes that facilitate its interaction with heterotrimeric G proteins, which then relay signals to downstream intracellular effectors. …”
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GPCR-Hippo Signaling in Cancer by Jiaqian Luo, Fa-Xing Yu

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GPCR_LigandClassify.py; a rigorous machine learning classifier for GPCR targeting compounds by Marawan Ahmed, Horia Jalily Hasani, Subha Kalyaanamoorthy, Khaled Barakat

“…These data points were retrieved from the GPCR-Ligand Association (GLASS) database. We have used diverse molecular featurization methods to describe the input molecules. …”
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Structural Insights into the Intrinsically Disordered GPCR C-Terminal Region, Major Actor in Arrestin-GPCR Interaction by Myriam Guillien, Assia Mouhand, Aurélie Fournet, Amandine Gontier, Aleix Martí Navia, Tiago N. Cordeiro, Frédéric Allemand, Aurélien Thureau, Jean-Louis Banères, Pau Bernadó, Nathalie Sibille

Subjects: “…GPCR…”
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Expanding the Concept of G Protein-Coupled Receptor (GPCR) Dimer Asymmetry towards GPCR-Interacting Proteins by Ralf Jockers, Pascal Maurice, Maud Kamal

Subjects: “…GPCR…”
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Probing GPCR Dimerization Using Peptides by Zara Farooq, Zara Farooq, Lesley A. Howell, Peter J. McCormick

Subjects: “…GPCR (G protein coupled receptor)…”
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Capturing Peptide–GPCR Interactions and Their Dynamics by Anette Kaiser, Irene Coin

Subjects: “…GPCR activation…”
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DEER Analysis of GPCR Conformational Heterogeneity by Matthias Elgeti, Wayne L. Hubbell

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Frequent substructure mining of GPCR ligands by IJzerman AP, Bender A, Horst E

Receptor-Arrestin Interactions: The GPCR Perspective by Mohammad Seyedabadi, Mehdi Gharghabi, Eugenia V. Gurevich, Vsevolod V. Gurevich

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Conformational dynamics in GPCR signaling by NMR by Yunfei Hu, Changwen Jin

Subjects: “…G-protein-coupled receptor (GPCR)…”
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Improved GPCR ligands from nanobody tethering by Ross W. Cheloha, Fabian A. Fischer, Andrew W. Woodham, Eileen Daley, Naomi Suminski, Thomas J. Gardella, Hidde L. Ploegh

“…Here the authors present a strategy for fusing nanobodies to suboptimal GPCR peptide ligands to potently and selectively activate receptors.…”
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Screening of GPCR drugs for repurposing in breast cancer by Noor Mazin Abdulkareem, Raksha Bhat, Reid T. Powell, Soumya Chikermane, Soham Yande, Lisa Trinh, Hala Y. Abdelnasser, Mantasha Tabassum, Alexis Ruiz, Mary Sobieski, Nghi D. Nguyen, Jun Hyoung Park, Camille A. Johnson, Benny A. Kaipparettu, Richard A. Bond, Michael Johnson, Clifford Stephan, Meghana V. Trivedi, Meghana V. Trivedi

“…In this study, we evaluated GPCR-targeting drugs by high throughput screening (HTS) for their repurposing potential in triple-negative breast cancer (TNBC) and drug-resistant human epidermal growth factor receptor-2-positive (HER2+) breast cancer (BC), due to the dire need to discover novel targets and drugs in these subtypes. …”
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GPCR Signaling Regulation: The Role of GRKs and Arrestins by Vsevolod V. Gurevich, Eugenia V. Gurevich

Subjects: “…GPCR…”
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Structural features of arrestin-mediated GPCR signaling by Wenqin Xie, Jinglin Lai, Hongmin Cai, H. Eric Xu, Wanchao Yin

Subjects: “…GPCR signalling…”
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A non-canonical mechanism of GPCR activation by Alexander S. Powers, Aasma Khan, Joseph M. Paggi, Naomi R. Latorraca, Sarah Souza, Jerry Di Salvo, Jun Lu, Stephen M. Soisson, Jennifer M. Johnston, Adam B. Weinglass, Ron O. Dror

“…Decades of research have led to the widely accepted view that all agonists—ligands that trigger GPCR activation—function by causing rearrangement of the GPCR’s transmembrane helices, opening an intracellular pocket for binding of transducer proteins. …”
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