Medicinal chemistry research progress / by Colombo, Giulia P., Ricci, Sofia

Discovery of the Orally Effective Thyrotropin-Releasing Hormone Mimetic: 1‑{N‑[(4S,5S)‑(5-Methyl-2-oxooxazolidine-4-yl)carbonyl]-3-(thiazol-4-yl)‑l‑alanyl}-(2R)‑2-methylpyrrolidine... by Naotake Kobayashi, Norihito Sato, Yuko Fujimura, Tsuyoshi Kihara, Katsuji Sugita, Kouji Takahashi, Katsumi Koike, Tamio Sugawara, Yukio Tada, Hiroshi Nakai, Takayoshi Yoshikawa

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The Corey-Seebach Reagent in the 21st Century: A Review by Muhammad Haroon, Ameer Fawad Zahoor, Sajjad Ahmad, Asim Mansha, Muhammad Irfan, Aqsa Mushtaq, Rabia Akhtar, Ali Irfan, Katarzyna Kotwica-Mojzych, Mariusz Mojzych

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Search for structurally diverse heterocyclic analogs as dual-acting antimalarial and antileishmanial agents: An overview by Faheem, Sanchita Dey, Samridhi Johri, M. Abirami, Banoth Karan Kumar, Donatella Taramelli, Nicoletta Basilico, Rafael Balana-Fouce, Kondapalli Venkata Gowri Chandra Sekhar, Sankaranarayanan Murugesan

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Simmons–Smith Cyclopropanation: A Multifaceted Synthetic Protocol toward the Synthesis of Natural Products and Drugs: A Review by Ramsha Munir, Ameer Fawad Zahoor, Sadia Javed, Bushra Parveen, Asim Mansha, Ahmad Irfan, Samreen Gul Khan, Ali Irfan, Katarzyna Kotwica-Mojzych, Mariusz Mojzych

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Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors by Péter Ábrányi-Balogh, Aaron Keeley, György G. Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast, Damijan Knez, Janez Ilaš, Stanislav Gobec, György M. Keserű

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Continuous-Flow Synthesis of Thioureas, Enabled by Aqueous Polysulfide Solution by András Gy. Németh, Renáta Szabó, György Orsy, István M. Mándity, György M. Keserű, Péter Ábrányi-Balogh

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Activation-Free Sulfonyl Fluoride Probes for Fragment Screening by László Petri, Péter Ábrányi-Balogh, Noémi Csorba, Aaron Keeley, József Simon, Ivan Ranđelović, József Tóvári, Gitta Schlosser, Dániel Szabó, László Drahos, György M. Keserű

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Similarity-based pairing improves efficiency of siamese neural networks for regression tasks and uncertainty quantification by Yumeng Zhang, Janosch Menke, Jiazhen He, Eva Nittinger, Christian Tyrchan, Oliver Koch, Hongtao Zhao

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Prediction of PPAR-α ligand-mediated physiological changes using gene expression profiles by Klaus Stensgaard Frederiksen, Erik Max Wulff, Per Sauerberg, John Patrick Mogensen, Lone Jeppesen, Jan Fleckner

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Implications of Additivity and Nonadditivity for Machine Learning and Deep Learning Models in Drug Design by Karolina Kwapien, Eva Nittinger, Jiazhen He, Christian Margreitter, Alexey Voronov, Christian Tyrchan

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Recent Trends in the Petasis Reaction: A Review of Novel Catalytic Synthetic Approaches with Applications of the Petasis Reaction by Sadaf Saeed, Saba Munawar, Sajjad Ahmad, Asim Mansha, Ameer Fawad Zahoor, Ali Irfan, Ahmad Irfan, Katarzyna Kotwica-Mojzych, Malgorzata Soroka, Mariola Głowacka, Mariusz Mojzych

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Design and Development of Small-Molecule Arylaldoxime/5-Nitroimidazole Hybrids as Potent Inhibitors of MARK4: A Promising Approach for Target-Based Cancer Therapy by Mudasir Nabi Peerzada, Parvez Khan, Nashrah Sharif Khan, Fernando Avecilla, Shadab Miyan Siddiqui, Md. Imtaiyaz Hassan, Amir Azam

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Chitosan-based films with cannabis oil as a base material for wound dressing application by Dorota Chelminiak-Dudkiewicz, Aleksander Smolarkiewicz-Wyczachowski, Kinga Mylkie, Magdalena Wujak, Dariusz T. Mlynarczyk, Pawel Nowak, Szymon Bocian, Tomasz Goslinski, Marta Ziegler-Borowska

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Sharpless Asymmetric Dihydroxylation: An Impressive Gadget for the Synthesis of Natural Products: A Review by Aqsa Mushtaq, Ameer Fawad Zahoor, Muhammad Bilal, Syed Makhdoom Hussain, Muhammad Irfan, Rabia Akhtar, Ali Irfan, Katarzyna Kotwica-Mojzych, Mariusz Mojzych

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Effect of Irradiation on Structural Changes of Levan by Dorota Chelminiak-Dudkiewicz, Aleksander Smolarkiewicz-Wyczachowski, Katarzyna Wegrzynowska-Drzymalska, Marta Ziegler-Borowska

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Pyridine- and Thiazole-Based Hydrazides with Promising Anti-inflammatory and Antimicrobial Activities along with Their In Silico Studies by Vinuta Kamat, Rangappa Santosh, Boja Poojary, Suresh P. Nayak, Banoth Karan Kumar, Murugesan Sankaranarayanan, Faheem, Sheela Khanapure, Delicia Avilla. Barretto, Shyam K. Vootla

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Late-stage synthesis of heterobifunctional molecules for PROTAC applications via ruthenium-catalysed C‒H amidation by Daniele Antermite, Stig D. Friis, Johan R. Johansson, Okky Dwichandra Putra, Lutz Ackermann, Magnus J. Johansson

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Discovery of Immunoproteasome Inhibitors Using Large-Scale Covalent Virtual Screening by Andrea Scarpino, Dávid Bajusz, Matic Proj, Martina Gobec, Izidor Sosič, Stanislav Gobec, György G. Ferenczy, György M. Keserű

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Sequence-based prediction of the intrinsic solubility of peptides containing non-natural amino acids by Marc Oeller, Ryan J. D. Kang, Hannah L. Bolt, Ana L. Gomes dos Santos, Annika Langborg Weinmann, Antonios Nikitidis, Pavol Zlatoidsky, Wu Su, Werngard Czechtizky, Leonardo De Maria, Pietro Sormanni, Michele Vendruscolo

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