Gel-Free Tools for Quick and Simple Screening of Anti-Topoisomerase 1 Compounds by Josephine Geertsen Keller, Kamilla Vandsø Petersen, Karol Mizielinski, Celine Thiesen, Lotte Bjergbæk, Rosa M. Reguera, Yolanda Pérez-Pertejo, Rafael Balaña-Fouce, Angela Trejo, Carme Masdeu, Concepcion Alonso, Birgitta R. Knudsen, Cinzia Tesauro

Subjects: “…human topoisomerase 1…”
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Bulge oligonucleotide as an inhibitory agent of bacterial topoisomerase I by Zhaoqi Yang, Tuoyu Jiang, Hanshi Zhong, Yu Kang

Subjects: “…Bacterial topoisomerase I…”
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Synthesis, DNA Binding and Topoisomerase I Inhibition Activity of Thiazacridine and Imidazacridine Derivatives by Elizabeth Almeida Lafayette, Sinara Mônica Vitalino de Almeida, Marina Galdino da Rocha Pitta, Eduardo Isidoro Carneiro Beltrão, Teresinha Gonçalves da Silva, Ricardo Olímpio de Moura, Ivan da Rocha Pitta, Luiz Bezerra de Carvalho, Maria do Carmo Alves de Lima

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Late onset systemic sclerosis with seronegativity: a rare presentation of an uncommon disease by D. Saxena, D. Jain, M. Yadav, K. Giri, T. Yadav, P. jain

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Pharmacokinetics and safety of DTS-108, a human oligopeptide bound to SN-38 with an esterase-sensitive cross-linker in patients with advanced malignancies: a Phase I study by Coriat R, Faivre SJ, Mir O, Dreyer C, Ropert S, Bouattour M, Desjardins R, Goldwasser F, Raymond E

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The combination of olaparib and camptothecin for effective radiosensitization by Miura Katsutoshi, Sakata Koh-ichi, Someya Masanori, Matsumoto Yoshihisa, Matsumoto Hideki, Takahashi Akihisa, Hareyama Masato

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Topoisomerase 1 Activity Is Reduced in Response to Thermal Stress in Fruit Flies and in Human HeLa Cells by Trine Juul-Kristensen, Josephine Geertsen Keller, Kathrine Nygaard Borg, Noriko Y. Hansen, Amalie Foldager, Rasmus Ladegaard, Yi-Ping Ho, Volker Loeschcke, Birgitta R. Knudsen

Subjects: “…topoisomerase 1…”
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Topoisomerase I in Human Disease Pathogenesis and Treatments by Min Li, Yilun Liu

Subjects: “…Topoisomerase 1…”
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Anti-Colorectal Cancer Effects of a Novel Camptothecin Derivative PCC0208037 <i>In Vitro</i> and <i>In Vivo</i> by Min Li, Linxu Wang, Yingjie Wei, Wenyan Wang, Zongliang Liu, Aixia Zuo, Wanhui Liu, Jingwei Tian, Hongbo Wang

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Mitochondrial topoisomerase 1 inhibition induces topological DNA damage and T cell dysfunction in patients with chronic viral infection by Xindi Dang, Xindi Dang, Dechao Cao, Dechao Cao, Juan Zhao, Juan Zhao, Madison Schank, Madison Schank, Sushant Khanal, Sushant Khanal, Lam Ngoc Thao Nguyen, Lam Ngoc Thao Nguyen, Xiao Y. Wu, Xiao Y. Wu, Yi Zhang, Yi Zhang, Jinyu Zhang, Jinyu Zhang, Yong Jiang, Yong Jiang, Shunbin Ning, Shunbin Ning, Ling Wang, Ling Wang, Mohamed El Gazzar, Mohamed El Gazzar, Jonathan P. Moorman, Jonathan P. Moorman, Jonathan P. Moorman, Zhi Q. Yao, Zhi Q. Yao, Zhi Q. Yao

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Non-Invasive Malaria Detection in Sub-Saharan Africa Using a DNA-Based Sensor System by Trine Juul-Kristensen, Celine Thiesen, Line Wulff Haurum, Josephine Geertsen Keller, Romeo Wenceslas Lendamba, Rella Zoleko Manego, Madeleine Eunice Betouke Ongwe, Birgitta Ruth Knudsen, Eduardo Pareja, Eduardo Pareja-Tobes, Rodrigo Labouriau, Ghyslain Mombo-Ngoma, Cinzia Tesauro

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Inhibitory effects of lapachol on rat C6 glioma in vitro and in vivo by targeting DNA topoisomerase I and topoisomerase II by Huanli Xu, Qunying Chen, Hong Wang, Pingxiang Xu, Ru Yuan, Xiaorong Li, Lu Bai, Ming Xue

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Dimethylmyricacene: An In Vitro and In Silico Study of a Semisynthetic Non-Camptothecin Derivative Compound, Targeting Human DNA Topoisomerase 1B by Alessio Ottaviani, Federico Iacovelli, Joshua Welsch, Blasco Morozzo della Rocca, Alessandro Desideri, Mattia Falconi, Laurent Calcul, Bill J. Baker, Paola Fiorani

Subjects: “…human topoisomerase 1B…”
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PHARMACOLOGIC TOPOISOMERASE-I INHIBITION CAUSES DNA DAMAGE AND MORTALITY IN ACTIVATED CD4+ T CELLS by Mia Stanić, Iart Luca Shytaj, Marina Lusic

Subjects: “…Topoisomerase-I…”
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Topoisomerase I prevents transcription-replication conflicts at transcription termination sites by Yaqun Liu, Yea-Lih Lin, Philippe Pasero, Chun-Long Chen

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Naturally Occurring Cytotoxic [3′→8″]-Biflavonoids from Podocarpus nakaii by Pen-Ho Yeh, Yun-Dar Shieh, Li-Chun Hsu, Li-Ming Yang Kuo, Jhih-Hu Lin, Chia-Ching Liaw, Yao-Haur Kuo

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Payload diversification: a key step in the development of antibody–drug conjugates by Louise Conilh, Lenka Sadilkova, Warren Viricel, Charles Dumontet

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Exatecan Antibody Drug Conjugates Based on a Hydrophilic Polysarcosine Drug-Linker Platform by Louise Conilh, Guy Fournet, Eric Fourmaux, Angélique Murcia, Eva-Laure Matera, Benoît Joseph, Charles Dumontet, Warren Viricel

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5,8-Dimethyl-9<i>H</i>-carbazole Derivatives Blocking hTopo I Activity and Actin Dynamics by Jessica Ceramella, Domenico Iacopetta, Anna Caruso, Annaluisa Mariconda, Anthi Petrou, Athina Geronikaki, Camillo Rosano, Carmela Saturnino, Alessia Catalano, Pasquale Longo, Maria Stefania Sinicropi

Subjects: “…human topoisomerases I/II…”
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Topoisomerase I inhibitor suppress tumor growth in chemoresistant ovarian cancer-initiating cells by Yu-Chi Wang, Cheng-Chang Chang, Kai-Jo Chiang, Tai-Kuang Chao, Chia-Chun Wu, Ping-Ying Chang, Chang-Chieh Wu, Hung-Cheng Lai

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