Solid-phase synthesis and biological evaluation of piperazine-based novel bacterial topoisomerase inhibitors by Flagstad, Thomas, Pedersen, Mette T., Jakobsen, Tim H., Felding, Jakob, Tolker-Nielsen, Tim, Givskov, Michael, Qvortrup, Katrine, Nielsen, Thomas E.

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SUMO: A Swiss Army Knife for Eukaryotic Topoisomerases by Yilun Sun, John L. Nitiss, Yves Pommier

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DNA topoisomerases as molecular targets for anticancer drugs by Kamila Buzun, Anna Bielawska, Krzysztof Bielawski, Agnieszka Gornowicz

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Determination of the Primary Molecular Target of 1,2,4-Triazole-Ciprofloxacin Hybrids by Tomasz Plech, Barbara Kaproń, Agata Paneth, Urszula Kosikowska, Anna Malm, Aleksandra Strzelczyk, Paweł Stączek, Łukasz Świątek, Barbara Rajtar, Małgorzata Polz-Dacewicz

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Design, synthesis and mechanistic study of N-4-Piperazinyl Butyryl Thiazolidinedione derivatives of ciprofloxacin with Anticancer Activity via Topoisomerase I/II inhibition by Hossameldin A. Aziz, Ahmed M. El-Saghier, Mohamed badr, Bakheet E. M. Elsadek, Gamal El-Din A. Abuo-Rahma, Mai E. Shoman

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Camptothecin bioprocessing from Aspergillus terreus, an endophyte of Catharanthus roseus: antiproliferative activity, topoisomerase inhibition and cell cycle analysis by Ashraf S. A. El-Sayed, Abdelaleim I. ElSayed, Khalid M. Wadan, Sayed S. El-Saadany, Nouran A. A. Abd El-Hady

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Bioprocessing of camptothecin from Alternaria brassicicola, an endophyte of Catharanthus roseus, with a strong antiproliferative activity and inhibition to Topoisomerases by Nouran A. A. Abd El-Hady, Abdelaleim I. ElSayed, Khalid M. Wadan, Sayed S. El-Saadany, Ashraf S. A. El-Sayed

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Topoisomerases inhibition and DNA binding mode of daunomycin–oligoarginine conjugate by Valeria Visone, Ildikó Szabó, Giuseppe Perugino, Ferenc Hudecz, Zoltán Bánóczi, Anna Valenti

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WHO HAS THERAPY-RELATED AML? by Robert Gale, John M. Bennett, F. Owen Hoffman

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Enhancing Antibacterial Efficacy: Combining Novel Bacterial Topoisomerase Inhibitors with Efflux Pump Inhibitors and Other Agents Against Gram-Negative Bacteria by Maša Zorman, Maja Kokot, Irena Zdovc, Lidija Senerovic, Mina Mandic, Nace Zidar, Andrej Emanuel Cotman, Martina Durcik, Lucija Peterlin Mašič, Nikola Minovski, Marko Anderluh, Martina Hrast Rambaher

Subjects: “…topoisomerase inhibitors…”
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Differential in vitro activity of the DNA topoisomerase inhibitor idarubicin against Trypanosoma rangeli and Trypanosoma cruzi by Momodou Jobe, Charles Anwuzia-Iwegbu, Ama Banful, Emma Bosier, Mubeen Iqbal, Kelly Jones, Suzanne J Lecutier, Kasimir Lepper, Matt Redmond, Andrew Ross-Parker, Emily Ward, Paul Wernham, Eleanor M Whidden, Kevin M Tyler, Dietmar Steverding

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A Fine-Tuned Lipophilicity/Hydrophilicity Ratio Governs Antibacterial Potency and Selectivity of Bifurcated Halogen Bond-Forming NBTIs by Anja Kolarič, Maja Kokot, Martina Hrast, Matjaž Weiss, Irena Zdovc, Jurij Trontelj, Simon Žakelj, Marko Anderluh, Nikola Minovski

Subjects: “…novel bacterial topoisomerase inhibitors…”
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The Implication of Topoisomerase II Inhibitors in Synthetic Lethality for Cancer Therapy by Victor M. Matias-Barrios, Xuesen Dong

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Topoisomerase inhibitors promote cancer cell motility via ROS-mediated activation of JAK2-STAT1-CXCL1 pathway by Jiafei Liu, Like Qu, Lin Meng, Chengchao Shou

Subjects: “…Topoisomerase inhibitors…”
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<i>In Vitro</i> Activity of Novel Topoisomerase Inhibitors against <i>Francisella tularensis</i> and <i>Burkholderia pseudomallei</i> by Adam O. Whelan, Ian Cooper, Nicola Ooi, David Orr, Kevin Blades, James Kirkham, Amanda Lyons, Kay B. Barnes, Mark I. Richards, Anne-Marie Salisbury, Mark Craighead, Sarah V. Harding

Subjects: “…topoisomerase inhibitors…”
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Special Issue “Anticancer Drugs” by Mary J. Meegan, Niamh M. O’Boyle

Subjects: “…conjugate and hybrid drugs, cisplatin resistance, topoisomerase inhibitors…”
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Topoisomerase Inhibitors Increase Episomal DNA Expression by Inducing the Integration of Episomal DNA in Hepatic Cells by Andoni Gómez-Moreno, Enara San Sebastian, Jennifer Moya, Pilar Gomollón-Zueco, Sergio Isola, África Vales, Gloria González-Aseguinolaza, Carmen Unzu, Urtzi Garaigorta

Subjects: “…topoisomerase inhibitor…”
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JNC-1043, a Novel Podophyllotoxin Derivative, Exerts Anticancer Drug and Radiosensitizer Effects in Colorectal Cancer Cells by Jin-Hee Kwon, Na-Gyeong Lee, A-Ram Kang, In-Ho Ahn, In-Young Choi, Jie-Young Song, Sang-Gu Hwang, Hong-Duck Um, Jong-Ryoo Choi, Joon Kim, Jong Kuk Park

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Antioxidant and antitopoisomerase activities in plant extracts of some Colombian flora from La Marcada Natural Regional Park by Jaime Niño, YanedMilena Correa, GermánDavid Cardona, Oscar Marino Mosquera

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The Aza-Analogous Benzo[<i>c</i>]phenanthridine P8-D6 Acts as a Dual Topoisomerase I and II Poison, thus Exhibiting Potent Genotoxic Properties by Georg Aichinger, Falk-Bach Lichtenberger, Tamara N. Steinhauer, Inken Flörkemeier, Giorgia Del Favero, Bernd Clement, Doris Marko

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