Docking, Binding Free Energy Calculations and In Vitro Characterization of Pyrazine Linked 2-Aminobenzamides as Novel Class I Histone Deacetylase (HDAC) Inhibitors by Emre F. Bülbül, Jelena Melesina, Hany S. Ibrahim, Mohamed Abdelsalam, Anita Vecchio, Dina Robaa, Matthes Zessin, Mike Schutkowski, Wolfgang Sippl

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Application of Ligand- and Structure-Based Prediction Models for the Design of Alkylhydrazide-Based HDAC3 Inhibitors as Novel Anti-Cancer Compounds by Emre F. Bülbül, Dina Robaa, Ping Sun, Fereshteh Mahmoudi, Jelena Melesina, Matthes Zessin, Mike Schutkowski, Wolfgang Sippl

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Synthesis, Molecular Docking and Biological Characterization of Pyrazine Linked 2-Aminobenzamides as New Class I Selective Histone Deacetylase (HDAC) Inhibitors with Anti-Leukemic... by Hany S. Ibrahim, Mohamed Abdelsalam, Yanira Zeyn, Matthes Zessin, Al-Hassan M. Mustafa, Marten A. Fischer, Patrik Zeyen, Ping Sun, Emre F. Bülbül, Anita Vecchio, Frank Erdmann, Matthias Schmidt, Dina Robaa, Cyril Barinka, Christophe Romier, Mike Schutkowski, Oliver H. Krämer, Wolfgang Sippl

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New Safety Aspects in Corneal Donation—Studies on SARS-CoV-2-Positive Corneal Donors by Diana Wille, Joana Heinzelmann, Astrid Kehlen, Marc Lütgehetmann, Dominik S. Nörz, Udo Siebolts, Anke Mueller, Matthias Karrasch, Nicola Hofmann, Anja Viestenz, Martin Börgel, Ferenc Kuhn, Arne Viestenz

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Betulin Sulfonamides as Carbonic Anhydrase Inhibitors and Anticancer Agents in Breast Cancer Cells by Antje Güttler, Yvonne Eiselt, Anne Funtan, Andreas Thiel, Marina Petrenko, Jacqueline Keßler, Iris Thondorf, Reinhard Paschke, Dirk Vordermark, Matthias Bache

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Design, Synthesis and Biological Characterization of Histone Deacetylase 8 (HDAC8) Proteolysis Targeting Chimeras (PROTACs) with Anti-Neuroblastoma Activity by Salma Darwish, Ehab Ghazy, Tino Heimburg, Daniel Herp, Patrik Zeyen, Rabia Salem-Altintas, Johannes Ridinger, Dina Robaa, Karin Schmidtkunz, Frank Erdmann, Matthias Schmidt, Christophe Romier, Manfred Jung, Ina Oehme, Wolfgang Sippl

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Binding Free Energy (BFE) Calculations and Quantitative Structure–Activity Relationship (QSAR) Analysis of <i>Schistosoma mansoni</i> Histone Deacetylase 8 (<i>sm</i>HDAC8) Inhibit... by Conrad V. Simoben, Ehab Ghazy, Patrik Zeyen, Salma Darwish, Matthias Schmidt, Christophe Romier, Dina Robaa, Wolfgang Sippl

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Repetitive Bleomycin-Based Electrochemotherapy Improves Antitumor Effectiveness in 3D Tumor Models of Conjunctival Melanoma by Joana Heinzelmann, Sabine Hecht, Alexander Ruben Vogt, Udo Siebolts, Peter Kaatzsch, Arne Viestenz

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Extracellular Acidosis Modulates the Expression of Epithelial-Mesenchymal Transition (EMT) Markers and Adhesion of Epithelial and Tumor Cells by Anne Riemann, Mandy Rauschner, Marina Gießelmann, Sarah Reime, Verena Haupt, Oliver Thews

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Complex Repetitive Discharges: A Sign of Motor Axonal Reinnervation? by Andreas Posa, Izabela Niśkiewicz, Alexander Emmer, Frank Hanisch, Malte E. Kornhuber

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<i>N</i>⁴-(2-Amino-4-fluorophenyl)-<i>N</i>¹-(3-{2-[2-(3-{[2-(2,6-dioxo-3-piperidyl)-1,3-dioxoisoindolin-4-yl]amino}propoxy)ethoxy]ethoxy}propyl)terephthalami... by Mohamed Abdelsalam, Matthes Zessin, Matthias Schmidt, Mike Schutkowski, Wolfgang Sippl

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The association of sleep patterns and depressive symptoms in medical students: a cross-sectional study by Katrin Dudo, Emilia Ehring, Stephan Fuchs, Sabine Herget, Stefan Watzke, Susanne Unverzagt, Thomas Frese

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The Conversion of Wollastonite to CaCO3 Considering Its Use for CCS Application as Cementitious Material by Kristoff Svensson, Andreas Neumann, Flora Feitosa Menezes, Christof Lempp, Herbert Pöllmann

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Elevated HERV-K Expression in Soft Tissue Sarcoma Is Associated with Worsened Relapse-Free Survival by Maria Giebler, Martin S. Staege, Sindy Blauschmidt, Lea I. Ohm, Matthias Kraus, Peter Würl, Helge Taubert, Thomas Greither

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Histone Deacetylase (HDAC) Inhibitors for the Treatment of Schistosomiasis by Ehab Ghazy, Mohamed Abdelsalam, Dina Robaa, Raymond J. Pierce, Wolfgang Sippl

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Phadiatop Seropositivity in Schizophrenia Patients and Controls: A Preliminary Study by Olaoluwa Okusaga, Robert G. Hamilton, Adem Can, Ajirioghene Igbide, Ina Giegling, Annette M. Hartmann, Bettina Konte, Marion Friedl, Gloria M Reeves, Dan Rujescu, Teodor T. Postolache

Investigation of Endogenous Retrovirus Sequences in the Neighborhood of Genes Up-regulated in a Neuroblastoma Model after Treatment with Hypoxia-Mimetic Cobalt Chloride by Christine Brütting, Christine Brütting, Harini Narasimhan, Frank Hoffmann, Malte E. Kornhuber, Martin S. Staege, Alexander Emmer

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Mason bees and honey bees synergistically enhance fruit set in sweet cherry orchards by Julia Osterman, Frances Benton, Sara Hellström, Meike Luderer‐Pflimpfl, Ann‐Kathrin Pöpel‐Eisenbrandt, Bilyana Stoykova Wild, Panagiotis Theodorou, Christin Ulbricht, Robert J. Paxton

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Role of advanced glycation end products in cellular signaling by Christiane Ott, Kathleen Jacobs, Elisa Haucke, Anne Navarrete Santos, Tilman Grune, Andreas Simm

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Comparative Structure-Based Virtual Screening Utilizing Optimized AlphaFold Model Identifies Selective HDAC11 Inhibitor by Fady Baselious, Sebastian Hilscher, Dina Robaa, Cyril Barinka, Mike Schutkowski, Wolfgang Sippl

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