Crystal structure of (2′,3,6′-trichlorobiphenyl-2-yl)boronic acid tetrahydrofuran monosolvate by Krzysztof Durka, Tomasz Kliś, Janusz Serwatowski

“…The title compound, C12H8BCl3O2·C4H8O, crystallizes as a tetrahydrofuran monosolvate. The boronic acid group adopts a syn–anti conformation and is significantly twisted along the carbon–boron bond by 69.2 (1)°, due to considerable steric hindrance from the 2′,6′-dichlorophenyl group that is located ortho to the boronic acid substituent. …”
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Cross-Linked Dependency of Boronic Acid-Conjugated Chitosan Nanoparticles by Diols for Sustained Insulin Release by Nabil A. Siddiqui, Nashiru Billa, Clive J. Roberts, Yaa Asantewaa Osei

“…Boronic acids have been widely investigated for their potential use as glucose sensors in glucose responsive polymeric insulin delivery systems. …”
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Development and Elucidation of a Novel Fluorescent Boron-Sensor for the Analysis of Boronic Acid-Containing Compounds by Yoshihide Hattori, Takuya Ogaki, Miki Ishimura, Yoichiro Ohta, Mitsunori Kirihata

“…Thus, in this paper, we report the development of a novel, convenient, and stable fluorescent boron-sensor based on O- and N-chelation (i.e., 2-(pyridine-2yl)phenol), and a corresponding method for the quantitative and qualitative detection of boronic acid-containing compounds using this commercially available sensor is presented.…”
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Responsive Boronic Acid-Decorated (Co)polymers: From Glucose Sensors to Autonomous Drug Delivery by Gertjan Vancoillie, Richard Hoogenboom

Subjects: “…boronic acid…”
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Simple Binding and Dissociation of a Sialoglycoprotein Using Boronic Acid-Modified Functional Interfaces on Microparticles by Yukichi Horiguchi, Masato Yasuura, Hiroki Ashiba, Zheng Lin Tan, Takashi Fukuda

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Group VIII metal carbonyl cluster-boronic acid conjugates : cytotoxicity and mode of action studies by Kong, Jia Wen, Lam, Zhiyong, Chan, Kiat Hwa, Ganguly, Rakesh, Lee, Joey Jia-Ying, Loo, Lit-Hsin, Webster, Richard D., Wong, Zhen Xuan, Leong, Weng Kee

“…A set of metal carbonyl cluster-boronic acid conjugates of the group VIII metals (Fe, Ru, and Os) were synthesized and their antiproliferative effects measured against two breast cancer cell lines (MCF-7 and MDA-MB-231) and a noncancerous breast epithelial (MCF-10A) cell line. …”
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Copper-Catalyzed Homocoupling of Boronic Acids: A Focus on B-to-Cu and Cu-to-Cu Transmetalations by Aude Salamé, Jordan Rio, Ilaria Ciofini, Lionel Perrin, Laurence Grimaud, Pierre-Adrien Payard

“…The presence of a coordinating base (hydroxide and methoxide) enables the B-to-Cu(II) transmetalation from aryl boronic acid to Cu^IICl₂ in methanol, through the formation of mixed Cu-(μ-OH)-B intermediates. …”
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Microwave-Assisted Regioselective Suzuki Coupling of 2,4-Dichloropyrimidines with Aryl and Heteroaryl Boronic Acids by Ana Dolšak, Kristjan Mrgole, Matej Sova

“…In this study, the Suzuki coupling of 2,4-dichloropyrimidines with aryl and heteroaryl boronic acids was investigated. A thorough screening of reaction conditions and the use of microwave irradiation led to a very efficient and straightforward synthetic procedure providing C4-substituted pyrimidines in good to excellent yields. …”
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Copper-mediated aerobic trifluoromethyltelluration of boronic acids with [Me4N][TeCF3] by Jing-Yan Dong, Hao-Nan Wang, Yan-Qian Xie, Cheng-Pan Zhang

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Dynamic combinatorial chemistry employing boronic acids/boronate esters leads to potent oxygenase inhibitors. by Demetriades, M, Leung, I, Chowdhury, R, Chan, M, McDonough, M, Yeoh, K, Tian, Y, Claridge, T, Ratcliffe, P, Woon, E, Schofield, C

“…Dynamic duo: The reversible reaction of boronic acids with alcohols to form boronate esters, coupled to protein mass spectrometry analyses, was used to discover potent oxygenase inhibitors. …”

Organoboronic acids/esters as effective drug and prodrug candidates in cancer treatments: challenge and hope by Mothana K. Al-Omari, Mai Elaarag, Raed M. Al-Zoubi, Ahmad R. Al-Qudimat, Ayman A. Zarour, Enas A. Al-Hurani, Zainab E. Fares, Leena M. Alkharraz, Mohanad Shkoor, Abdulilah D. Bani-Yaseen, Omar M. Aboumarzouk, Aksam Yassin, Abdulla A. Al-Ansari

Subjects: “…Boronic acid…”
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Boronic acid-functionalized tungsten disulfide quantum dots as a fluorescence probe for sensitive detection of dopamine by Rashmita Devi, Satyabrat Gogoi, Hemant Sankar Dutta, Prakash Jyoti Saikia, Ayushi Singhal, Raju Khan

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Oxidative Hydroxylation of Aryl Boronic Acid Catalyzed by Co-porphyrin Complexes via Blue-Light Irradiation by Alaa A. Atia, Masanari Kimura

Subjects: “…aryl boronic acid…”
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A boronic-acid-based probe for fluorescence polarization assays with penicillin binding proteins and β-lactamases by Inglis, SR, Strieker, M, Rydzik, A, Dessen, A, Schofield, C

A boronic-acid-based probe for fluorescence polarization assays with penicillin binding proteins and β-lactamases. by Inglis, SR, Strieker, M, Rydzik, A, Dessen, A, Schofield, C

“…We report the development of a fluorescence polarization (FP) assay for PBPs and "serine" β-lactamases using a boronic-acid-based, reversibly binding "tracer." The tracer was designed based on a crystal structure of a covalent complex between a boronic acid and PBP1b from Streptococcus pneumoniae. …”

Advancing Glycan Analysis: A New Platform Integrating SERS, Boronic Acids, and Machine Learning Algorithms by Qiang Hu, Dacheng Kuai, Hyundo Park, Haley Clark, Perla B. Balbuena, Joseph Sang‐Il Kwon, Hung‐Jen Wu

Subjects: “…boronic acids…”
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Copper-Catalyzed <i>N</i>-Arylation of Pyranoquinolinones with Boronic Acids at Room Temperature without Ligand by Wei Gao, Fang Gao, Haikuan Yang, Zongde Wang, Yaru Huang

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Boronic Acids of Pharmaceutical Importance Affect the Growth and Photosynthetic Apparatus of Cyanobacteria in a Dose-Dependent Manner by Emilia Niemczyk, Jerzy Pogrzeba, Agnieszka Adamczyk-Woźniak, Jacek Lipok

Subjects: “…aryl boronic acids…”
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Synthesis of 18F-difluoromethylarenes using aryl boronic acids, ethyl bromofluoroacetate and [18F]fluoride by Sap, J, Wilson, T, Kee, C, Straathof, N, Ende, C, Mukherjee, P, Zhang, L, Genicot, C, Gouverneur, V

Efficient pH-Responsive Nano-Drug Delivery System Based on Dynamic Boronic Acid/Ester Transformation by Weijun Chen, Wanxuan Xie, Guangkuo Zhao, Qi Shuai

“…To address this issue, we designed and prepared a boronic acid/ester-based pH-responsive nano-drug delivery system that targets the acidic microenvironment of tumors. …”
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