Regioselective alkynylation followed by Suzuki coupling of 2,4-dichloroquinoline: Synthesis of 2-alkynyl-4-arylquinolines by Ellanki A. Reddy, Aminul Islam, K. Mukkanti, Venkanna Bandameedi, Dipal R. Bhowmik, Manojit Pal

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Synthesis of Paclitaxel Derivatives for Remote Loading into Liposomes and Improved Therapeutic Effect by Xiangwei Xu, Yanhua Liu, Shanshan Shao, Jinbo Li, Zhaochu Xu, Yueling Yin, Linxiang Zhao, Yongjun Wang, Dan Liu

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2′-Chloro-4-(1-methyl-1H-imidazol-2-yl)-2,4′-bipyridine by Dhafer Saber Zinad, Dunya L. AL-Duhaidahaw, Ahmed Al-Amiery

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Fulvestrant-3-Boronic Acid (ZB716) Demonstrates Oral Bioavailability and Favorable Pharmacokinetic Profile in Preclinical ADME Studies by Jiawang Liu, Nirmal Rajasekaran, Ahamed Hossain, Changde Zhang, Shanchun Guo, Borui Kang, Hunsoon Jung, Hongjoong Kim, Guangdi Wang

“…Fulvestrant-3-boronic acid (ZB716), an oral selective estrogen receptor degrader (SERD) under clinical development, has been investigated in ADME studies to characterize its absorption, metabolism, and pharmacokinetics. …”
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Structural analysis of the boronic acid β-lactamase inhibitor vaborbactam binding to Pseudomonas aeruginosa penicillin-binding protein 3 by Vijay Kumar, Samantha L. Viviani, Jeeda Ismail, Shreya Agarwal, Robert A. Bonomo, Focco van den Akker

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Structural analysis of the boronic acid β-lactamase inhibitor vaborbactam binding to Pseudomonas aeruginosa penicillin-binding protein 3. by Vijay Kumar, Samantha L Viviani, Jeeda Ismail, Shreya Agarwal, Robert A Bonomo, Focco van den Akker

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Detection and first characterization of an uncommon haptoglobin in porcine saliva of pigs with rectal prolapse by using boronic acid sample enrichment by A.M. Gutiérrez, I. Miller, D. Kolarich, K. Hummel, K. Nöbauer, E. Razzazi-Fazeli

“…Salivary glycoprotein profiles, obtained after boronic acid enrichment, were studied for the first time in pigs in order to search for specific overall alterations related to acute inflammatory condition. …”
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Phenylboronic Acid-Functionalized Micelles Dual-Targeting Boronic Acid Transporter and Polysaccharides for siRNA Delivery into Brown Algae by Naoto Yoshinaga, Takaaki Miyamoto, Mami Goto, Atsuko Tanaka, Keiji Numata

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Facile Fabrication of Hierarchically Porous Boronic Acid Group-Functionalized Monoliths With Optical Activity for Recognizing Glucose With Different Conformation by Yan Wang, Luwei Zhang, Yu-I Hsu, Taka-Aki Asoh, Hiroshi Uyama

“…In particular, the boronic acid functional group that can interact with a cis-diol group was successfully introduced on the skeleton surface of the monoliths. …”
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Reactive Extraction Of Sugars From Oil Palm Empty Fruit Bunch Hydrolysate Using Naphthalene-2-Boronic Acid. by Abdul Aziz, Hanida

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A convenient catalyst system for microwave accelerated cross-coupling of a range of aryl boronic acids with aryl chlorides by Matthew L. Clarke, Marcia B. France, Jose A. Fuentes, Edward J. Milton, Geoffrey J. Roff

“…A convenient microwave accelerated cross-coupling procedure between aryl chlorides with a range of boronic acids has been developed. An explanation for the low reactivity of highly fluorinated boronic acids in Suzuki coupling is provided.…”
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Active Palladium Colloids via Palladacycle Degradation as Efficient Catalysts for Oxidative Homocoupling and Cross-Coupling of Aryl Boronic Acids by Vaibhav Sable, Karan Maindan, Anant R. Kapdi, Pushkar Sudhakar Shejwalkar, Kenji Hara

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Copper-Catalyzed Synthesis of Unsymmetrical Diorganyl Chalcogenides (Te/Se/S) from Boronic Acids under Solvent-Free Conditions by Sumbal Saba, Giancarlo Vaccari Botteselle, Marcelo Godoi, Tiago Elias Allievi Frizon, Fábio Zazyki Galetto, Jamal Rafique, Antonio L. Braga

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Synthesis of aryldifluoromethyl aryl ethers via nickel-catalyzed suzuki cross-coupling between aryloxydifluoromethyl bromides and boronic acids by Heng Lu, Ruo-Xuan Xiao, Chang-Yun Shi, Zi-Lan Song, Hou-Wen Lin, Ao Zhang

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Crown Ether-Derived Chiral BINOL: Enantioselective Michael Addition of Alkenyl Boronic Acids to α,β-Unsaturated Ketones by Jia-Ju Tao, Jia-Dong Tang, Tao Hong, Jia-Wen Ye, Jia-Yu Chen, Chunsong Xie, Zibin Zhang, Shijun Li

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Generating Selective Saccharide Binding Affinity of Phenyl Boronic Acids by using Single-Walled Carbon Nanotube Corona Phases by Mu, Bin, Ahn, Jiyoung, McNicholas, Thomas P., Strano, Michael S.

“…Herein, we demonstrate that a polymer or surfactant corona phase surrounding a single-walled carbon nanotube can substantially modify the selectivity of pre-adsorbed phenyl-boronic acids (PBA) for mono-, di-, and poly-saccharides. …”
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Carbon-carbon bond construction using boronic acids and aryl methyl sulfides: orthogonal reactivity in Suzuki-type couplings by Hooper, J, Young, R, Pernik, I, Weller, A, Willis, M

“…The Rh(i)-catalysed coupling of aryl and alkenyl boronic acids with simple aryl and alkenyl methyl sulfides is reported. …”

Palladium(II)-catalyzed synthesis of sulfinates from boronic acids and DABSO: a redox-neutral, phosphine-free transformation by Deeming, AS, Russell, CJ, Willis, MC

“…A redox-neutral palladium(II)-catalyzed conversion of aryl, heteroaryl, and alkenyl boronic acids into sulfinate intermediates, and onwards to sulfones and sulfonamides, has been realized. …”

SYNTHESIS AND CYTOTOXIC ACTIVITY OF 2,5-BIS(4-BORONIC ACID)BENZYLIDINE CYCLOPENTANONE ON HER2 OVEREXPRESSED-CANCER CELLS by Rohmad Yudi Utomo, Herwandhani Putri, Pudjono, Ratna Asmah Susidarti, Riris Istighfari Jenie, Edy Meiyanto

“…The purpose of this study is to synthesize curcumin analogue, namely Pentagamaboron-0 (PGB-0) or 2,5-bis(4-boronic acid)benzylidine cyclopentanone, and to explore the cytotoxic activity on HER2 overexpressed-cancer cells. …”
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Development of a method for the synthesis of 2,4,5-trisubstituted oxazoles composed of carboxylic acid, amino acid, and boronic acid by Kohei Yamada, Naoto Kamimura, Munetaka Kunishima

“…One-pot formation of 5-(triazinyloxy)oxazoles using carboxylic acids, amino acids and a dehydrative condensing reagent, DMT-MM, followed by Ni-catalyzed Suzuki–Miyaura coupling with boronic acids provided the corresponding 2,4,5-trisubstituted oxazoles in good yields.…”
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