X-ray Structure Determination, Antioxidant Voltammetry Studies of Butein and 2′,4′-Dihydroxy-3,4-dimethoxychalcone. Computational Studies of 4 Structurally Related 2′,4′-diOH Chalc... by Ijeoma Okoye, Sandra Yu, Francesco Caruso, Miriam Rossi

Subjects: “…falcipain-2…”
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Antimalarial dihydrochalcone isolated from Artocarpus sericicarpus Jarret leaves and in silico investigation against falcipain-2 protein by Lidya Tumewu, Hilkatul Ilmi, Ratih Dewi Saputri, Defi Kartika Sari, Adita Ayu Permanasari, Hanifah Khairun Nisa, Saipul Maulana, Tjitjik Srie Tjahjandarie, Mulyadi Tanjung, Che Puteh Osman, Nor Hadiani Ismail, Aty Widyawaruyanti, Achmad Fuad Hafid

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Design, synthesis, conformational and molecular docking study of some novel acyl hydrazone based molecular hybrids as antimalarial and antimicrobial agents by Parvin Kumar, Kulbir Kadyan, Meenakshi Duhan, Jayant Sindhu, Vineeta Singh, Baljeet Singh Saharan

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Novel series of 1,2,4-trioxane derivatives as antimalarial agents by Mithun Rudrapal, Dipak Chetia, Vineeta Singh

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Noscapine shows antimalarial activity against Plasmodium falciparum 3D7, its clinical isolate Pf140/SS, and Plasmodium berghei ANKA by Swaraj Kumar Babu, Sameer Maharana, Satyaranjan Chhatria, Dibya Ranjan Sahoo, Ashirbad Nanda, Satish Kanhar, Prativa K. Behera, Sanjib Mohanty, Pradeep Kumar Naik, Praveen Kishore Sahu

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In silico Guided Drug Repurposing: Discovery of New Competitive and Non-competitive Inhibitors of Falcipain-2 by Lucas N. Alberca, Sara R. Chuguransky, Cora L. Álvarez, Alan Talevi, Emir Salas-Sarduy

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Synthesis and Antimalarial Activity of Novel Dihydro-Artemisinin Derivatives by Jian Wang, Jin Huang, Chun Guo, Wei Luo, Yang Liu, Weiqiang Lu, Kunqiang Cui

Subjects: “…falcipain-2 inhibitors…”
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Virtual design of novel Plasmodium falciparum cysteine protease falcipain-2 hybrid lactone–chalcone and isatin–chalcone inhibitors probing the S2 active site pocket by Koffi N’Guessan Placide Gabin Allangba, Mélalie Keita, Raymond Kre N’Guessan, Eugene Megnassan, Vladimir Frecer, Stanislav Miertus

Subjects: “…falcipain-2…”
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2-Amido-3-(1H-Indol-3-yl)-N-Substitued-Propanamides as a New Class of Falcipain-2 Inhibitors. 1. Design, Synthesis, Biological Evaluation and Binding Model Studies by Tong Chen, Jin Zhu, Peng Che, Lili Chen, Weiqiang Lu, Jin Huang, Jian Li, Honglin Li, Hualiang Jiang

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Successful application of virtual screening and molecular dynamics simulations against antimalarial molecular targets by Renata Rachide Nunes, Marina dos Santos Costa, Bianca dos Reis Santos, Amanda Luisa da Fonseca, Lorena Sales Ferreira, Rafael Cesar Russo Chagas, Alisson Marques da Silva, Fernando de Pilla Varotti, Alex Gutterres Taranto

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Identification of Tight-Binding Plasmepsin II and Falcipain 2 Inhibitors in Aqueous Extracts of Marine Invertebrates by the Combination of Enzymatic and Interaction-Based Assays by Emir Salas-Sarduy, Yasel Guerra, Giovanni Covaleda Cortés, Francesc Xavier Avilés, María A. Chávez Planes

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Rational drug design, synthesis, and biological evaluation of novel N-(2-arylaminophenyl)-2,3-diphenylquinoxaline-6-sulfonamides as potential antimalarial, antifungal, and antibact... by Ahmed Hassen Shntaif, Sharuk Khan, Ganesh Tapadiya, Anand Chettupalli, Shweta Saboo, Mohd Sayeed Shaikh, Falak Siddiqui, Ramkoteswra Rao Amara

Subjects: “…Plasmodium cysteine protease falcipain-2…”
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Design, molecular docking, drug-likeness, and molecular dynamics studies of 1,2,4-trioxane derivatives as novel Plasmodium falciparum falcipain-2 (FP-2) inhibitors by Subham Ghosh, Dipak Chetia, Neelutpal Gogoi, Mithun Rudrapal

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2-(3,4-Dihydro-4-Oxothieno[2,3-d]pyrimidin-2-ylthio) Acetamides as a New Class of Falcipain-2 Inhibitors. 3. Design, Synthesis and Biological Evaluation by Hualiang Jiang, Jian Li, Honglin Li, Jin Huang, Weiqiang Lu, Ruoqun Ma, Jie Liu, Jin Zhu, Tong Chen

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A Novel Series of [1,2,4]Triazolo[4,3-a]Pyridine Sulfonamides as Potential Antimalarial Agents: In Silico Studies, Synthesis and In Vitro Evaluation by Veronika R. Karpina, Svitlana S. Kovalenko, Sergiy M. Kovalenko, Oleksandr G. Drushlyak, Natalya D. Bunyatyan, Victoriya A. Georgiyants, Vladimir V. Ivanov, Thierry Langer, Louis Maes

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