(E)-7-Ethylidene-lithocholic Acid (7-ELCA) Is a Potent Dual Farnesoid X Receptor (FXR) Antagonist and GPBAR1 Agonist Inhibiting FXR-Induced Gene Expression in Hepatocytes and Stimu... by Alzbeta Stefela, Miroslav Kaspar, Miroslav Kaspar, Martin Drastik, Thales Kronenberger, Thales Kronenberger, Stanislav Micuda, Martin Dracinsky, Blanka Klepetarova, Eva Kudova, Petr Pavek

Subjects: “…G protein-coupled bile acid receptor 1…”
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Bile acid activated receptors: Integrating immune and metabolic regulation in non-alcoholic fatty liver disease by Michele Biagioli, Stefano Fiorucci

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G protein-coupled bile acid receptor 1 activation attenuates endothelin-1-induced rat cardiomyocyte hypertrophy by inhibiting CaN/NAFT3 pathway by CHEN Dexiu, LI Jiafu, FENG Jian

Subjects: “…g protein-coupled bile acid receptor 1…”
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Intestinal flora and bile acid interactions impact the progression of diabetic kidney disease by Jia Xu, Nan Wang, Li Yang, Jing Zhong, Ming Chen

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Discovery of a Potent and Orally Active Dual GPBAR1/CysLT1R Modulator for the Treatment of Metabolic Fatty Liver Disease by Stefano Fiorucci, Pasquale Rapacciuolo, Bianca Fiorillo, Rosalinda Roselli, Silvia Marchianò, Cristina Di Giorgio, Martina Bordoni, Rachele Bellini, Chiara Cassiano, Paolo Conflitti, Bruno Catalanotti, Vittorio Limongelli, Vittorio Limongelli, Valentina Sepe, Michele Biagioli, Angela Zampella

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