Team-based learning-adopted strategy in pharmacy education: pharmacology and medicinal chemistry students’ perceptions by Reem T. Attia, Asmaa A. Mandour

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Heteroleptic Copper(I)-Based Complexes Incorporating BINAP and π-Extended Diimines: Synthesis, Catalysis and Biological Applications by Corentin Cruché, Sayak Gupta, Jeremy Kodanko, Shawn K. Collins

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Development of chemical tools to probe the functions of TRIM proteins by Reynolds, J

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Targeting the Ras superfamily via their regulatory GEF complexes by Gray, J

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Characterisation of novel evasins by Eaton, J

Subjects: “…Medicinal Chemistry…”

Boronic acid and nitrofuranyl derivatives as potential therapeutics by Dey, AL

Subjects: “…Medicinal Chemistry…”

Mutate & conjugate: a method for rapid in-cell validation of epigenetic targets by Thomas, AM

Subjects: “…Medicinal chemistry…”

Mechanisms underlying statin-induced modulation of ryanodine receptors by Lindsay, C

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Experimental biological studies of novel tetradentate hydrazone Cu(II) complexes for potential applications in medicinal chemistry by Cansu Topkaya

“…The obtained results highlight the significance of these novel complexes in the field of medicinal chemistry. …”
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From Medicinal Chemistry to Human Health: Current Approaches to Drug Discovery for Cancer and Neglected Tropical Diseases by LEONARDO G. FERREIRA, GLAUCIUS OLIVA, ADRIANO D. ANDRICOPULO

Subjects: “…medicinal chemistry…”
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Contemporary medicinal chemistry strategies for the discovery and optimization of influenza inhibitors targeting vRNP constituent proteins by Lingxin Hou, Ying Zhang, Han Ju, Srinivasulu Cherukupalli, Ruifang Jia, Jian Zhang, Bing Huang, Arianna Loregian, Xinyong Liu, Peng Zhan

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Pharmacokinetics-Driven Evaluation of the Antioxidant Activity of Curcuminoids and Their Major Reduced Metabolites—A Medicinal Chemistry Approach by Gábor Girst, Sándor B. Ötvös, Ferenc Fülöp, György T. Balogh, Attila Hunyadi

“…In this work, we aimed to perform a comparative evaluation of curcuminoids and their hydrogenated metabolites from a medicinal chemistry point of view, by determining a set of key pharmacokinetic parameters and evaluating antioxidant potential in relation to such properties.Reduced metabolites were prepared from curcumin and demethoxycurcumin through continuous-flow hydrogenation. …”
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Química Medicinal Moderna: desafios e contribuição brasileira Modern Medicinal Chemistry: challenges and Brazilian contribution by Lídia M. Lima

Subjects: “…medicinal chemistry…”
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Medicinal chemistry strategies towards the development of non-covalent SARS-CoV-2 Mpro inhibitors by Letian Song, Shenghua Gao, Bing Ye, Mianling Yang, Yusen Cheng, Dongwei Kang, Fan Yi, Jin-Peng Sun, Luis Menéndez-Arias, Johan Neyts, Xinyong Liu, Peng Zhan

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From Plant to Chemistry: Sources of Antinociceptive Non-Opioid Active Principles for Medicinal Chemistry and Drug Design by Rita Turnaturi, Silvia Piana, Salvatore Spoto, Giuliana Costanzo, Lorena Reina, Lorella Pasquinucci, Carmela Parenti

“…As the process of pain transmission and modulation is regulated by different peripheral and central mechanisms and neurotransmitters, medicinal chemistry continues to study novel ligands and innovative approaches. …”
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New dimensions in triazolo[4,3-a]pyrazine derivatives: The land of opportunity in organic and medicinal chemistry by Divya J. Jethava, Mayuri A. Borad, Manoj N. Bhoi, Prachi T. Acharya, Zeel A. Bhavsar, Hitesh D. Patel

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Assessing the impact of clinically relevant medicinal chemistry teaching: Learning gains from case study approach by Fernanda Domingues Lustoza, João Paulo S. Fernandes

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Exploring the structural and functional requirements of Phyto-compounds and their synthetic scaffolds as anticancer agents: Medicinal chemistry perspective by Dipanjan Karati, Dileep Kumar

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Chemical Upcycling of Expired Pharmaceuticals as a Source of Value-Added Chemicals for Organic Synthesis and Medicinal Chemistry by Teresa Abad-Grillo, Grant McNaughton-Smith

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Selective inhibitors of protozoan protein N-myristoyltransferases as starting points for tropical disease medicinal chemistry programs. by Andrew S Bell, James E Mills, Gareth P Williams, James A Brannigan, Anthony J Wilkinson, Tanya Parkinson, Robin J Leatherbarrow, Edward W Tate, Anthony A Holder, Deborah F Smith

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