Search for structurally diverse heterocyclic analogs as dual-acting antimalarial and antileishmanial agents: An overview by Faheem, Sanchita Dey, Samridhi Johri, M. Abirami, Banoth Karan Kumar, Donatella Taramelli, Nicoletta Basilico, Rafael Balana-Fouce, Kondapalli Venkata Gowri Chandra Sekhar, Sankaranarayanan Murugesan

“…European Journal of Medicinal Chemistry Reports…”
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Replacing the phthalimide core in thalidomide with benzotriazole by Mikhail Krasavin, Andrey Bubyrev, Alexander Kazantsev, Christopher Heim, Samuel Maiwald, Daniil Zhukovsky, Dmitry Dar’in, Marcus D. Hartmann, Alexander Bunev

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Tumor necrosis factor alpha (TNFα)-binding imprinted polymers. A non-systemic therapeutic approach for inflammatory bowel diseases by Rina Arad Yellin, Anett Hudák, Tamás Letoha, Bernard S. Green

“…European Journal of Medicinal Chemistry Reports…”
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Probing the role of an invariant active site His in family GH1 β-glycosidases by Andrea Strazzulli, Giuseppe Perugino, Marialuisa Mazzone, Mosè Rossi, Stephen G. Withers, Marco Moracci

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Seeking new approach for therapeutic treatment of cholera disease via inhibition of bacterial carbonic anhydrases: experimental and theoretical studies for sixteen benzenesulfonami... by Rosaria Gitto, Laura De Luca, Francesca Mancuso, Sonia Del Prete, Daniela Vullo, Claudiu T. Supuran, Clemente Capasso

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Targeting bacterial growth in biofilm conditions: rational design of novel inhibitors to mitigate clinical and food contamination using QSAR by Maria Galvez-Llompart, Jesús Hierrezuelo, Mariluz Blasco, Riccardo Zanni, Jorge Galvez, Antonio de Vicente, Alejandro Pérez-García, Diego Romero

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Portulaca oleracea leave extract enhanced renal function via enhancing urea and creatinine clearance in wistar rats by Naiho Alexander Obidike, Emojevwe Victor, Oyovwi Mega Obukohwo, Ohwin Peggy Ejiro, Osamah Ngozi Blessing

“…European Journal of Medicinal Chemistry Reports…”
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Correction to: Zhang et al., Discovery of novel PDE9A inhibitors with antioxidant activities for treatment of Alzheimer’s disease

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Differential expression of snoRNAs in oral squamous cell carcinomas: new potential diagnostic markers by Cintia Chamorro-Petronacci, Mario Perez-Sayáns, Maria Elena Padín-Iruegas, Xabier Marichalar-Mendia, Mercedes Gallas-Torreira, Abel García García

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Flavonoid-liposomes formulations: Physico-chemical characteristics, biological activities and therapeutic applications by Eleftherios G. Halevas, Dimitrios I. Avgoulas, George Katsipis, Anastasia A. Pantazaki

“…European Journal of Medicinal Chemistry Reports…”
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Design and green synthesis of novel quinolinone derivatives of potential anti-breast cancer activity against MCF-7 cell line targeting multi-receptor tyrosine kinases by Mohamed Mokhtar, Khadijah S. Alghamdi, Nesreen S. Ahmed, Dina Bakhotmah, Tamer S. Saleh

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Experimental modelling of Alzheimer's disease for therapeutic screening by Laura Blaikie, Graeme Kay, Patricia Maciel, Paul Kong Thoo Lin

“…European Journal of Medicinal Chemistry Reports…”
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Dependence on linkers’ flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents by Haytham O. Tawfik, Amany Belal, Mohammed A. S. Abourehab, Andrea Angeli, Alessandro Bonardi, Claudiu T. Supuran, Mervat H. El-Hamamsy

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Synthesis and antitumor activity of novel 2, 3-didithiocarbamate substituted naphthoquinones as inhibitors of pyruvate kinase M2 isoform by Xianling Ning, Hailong Qi, Ridong Li, Yan Jin, Michael A. McNutt, Yuxin Yin

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Design, synthesis, and evaluation of novel O-alkyl ferulamide derivatives as multifunctional ligands for treating Alzheimer’s disease by Gaofeng Zhu, Ping Bai, Keren Wang, Jing Mi, Jing Yang, Jiaqi Hu, Yujuan Ban, Ran Xu, Rui Chen, Changning Wang, Lei Tang, Zhipei Sang

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Designing, synthesis and bioactivities of 4-[3-(4-hydroxyphenyl)-5-aryl-4,5-dihydro-pyrazol-1-yl]benzenesulfonamides by Halise Inci Gul, Ebru Mete, Sakip Emre Eren, Hiroshi Sakagami, Cem Yamali, Claudiu T. Supuran

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Computer-aided design and synthesis of 3-carbonyl-5-phenyl-1H-pyrazole as highly selective and potent BRAFV600E and CRAF inhibitor by Jinwoong Kim, Byeongha Choi, Daseul Im, Hoyong Jung, Hyungwoo Moon, Waqar Aman, Jung-Mi Hah

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Thioredoxin-dependent system. Application of inhibitors by Anna Jastrząb, Elżbieta Skrzydlewska

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Hyperbaric oxygen therapy modulates serum OPG/RANKL in femoral head necrosis patients by Giuliano Vezzani, Silvia Quartesan, Pasqua Cancellara, Enrico Camporesi, Devanand Mangar, Thomas Bernasek, Prachiti Dalvi, Zhongjin Yang, Antonio Paoli, Alex Rizzato, Gerardo Bosco

“…Journal of Enzyme Inhibition and Medicinal Chemistry…”
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Recent advances on anticancer activity of coumarin derivatives by Anjali Rawat, A. Vijaya Bhaskar Reddy

“…European Journal of Medicinal Chemistry Reports…”
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