Medicinal Chemistry and Chemical Biology: Abstracts MC001-MC100

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A mini review on pyridoacridines: Prospective lead compounds in medicinal chemistry by Vikas Sharma, Prabodh C. Sharma, Vipin Kumar

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Immobilized artificial membrane chromatography: from medicinal chemistry to environmental sciences by Fotis Tsopelas, Chrysanthos Stergiopoulos, Anna Tsantili-Kakoulidou

“…The promising results in both medicinal chemistry and in environmental science in combination with the speed, reproducibility and low analyte consumption suggest that a broader application of IAM chromatography in the early drug discovery process and in ecotoxicity may save time and money in initial drug candidate selection and will contribute to a reduced risk hazard of chemicals.…”
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Small molecule angiotensin converting enzyme inhibitors: A medicinal chemistry perspective by Wenyue Zheng, Wenyue Zheng, Erkang Tian, Zhen Liu, Changhan Zhou, Pei Yang, Pei Yang, Keyue Tian, Wen Liao, Juan Li, Changyu Ren

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Imidazole: Synthesis, Functionalization and Physicochemical Properties of a Privileged Structure in Medicinal Chemistry by Heber Victor Tolomeu, Carlos Alberto Manssour Fraga

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3-Phenylcoumarins as a Privileged Scaffold in Medicinal Chemistry: The Landmarks of the Past Decade by Maria J. Matos, Eugenio Uriarte, Lourdes Santana

“…3-Phenylcoumarins are a family of heterocyclic molecules that are widely used in both organic and medicinal chemistry. In this overview, research on this scaffold, since 2010, is included and discussed, focusing on aspects related to its natural origin, synthetic procedures and pharmacological applications. …”
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Structural Characterization of 4-(4-Nitrophenyl)thiomorpholine, a Precursor in Medicinal Chemistry by Paul R. Palme, Richard Goddard, Peter Imming, Rüdiger W. Seidel

“…4-(4-nitrophenyl)thiomorpholine, the title compound, has been used as a precursor for the corresponding 4-thiomorpholinoaniline, which is a useful building block in medicinal chemistry. The crystal and molecular structures of the title compound, however, have not been described thus far. …”
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Thiopyrano[2,3-d]Thiazoles as New Efficient Scaffolds in Medicinal Chemistry by Anna Kryshchyshyn, Olexandra Roman, Andrii Lozynskyi, Roman Lesyk

“…Thiazolidine and thiazolidinone-related compounds belong to the widely studied heterocycles from a medicinal chemistry perspective. From the chemical point of view, they are perfect heterodienes to undergo hetero-Diels–Alder reaction with a variety of dienophiles, yielding regio- and diastereoselectively thiopyranothiazole scaffolds. …”
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Ion Channels and Transporters as Therapeutic Agents: From Biomolecules to Supramolecular Medicinal Chemistry by Giacomo Picci, Silvia Marchesan, Claudia Caltagirone

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Medicinal Chemistry of Annonaceous Acetogenins: Design, Synthesis, and Biological Evaluation of Novel Analogues by Naoto Kojima, Tetsuaki Tanaka

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The Combination of Solid-State Chemistry and Medicinal Chemistry as the Basis for the Synthesis of Theranostics Platforms by Dmitry Korolev, Viktor Postnov, Ilia Aleksandrov, Igor Murin

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Endocannabinoid Degradation Enzyme Inhibitors as Potential Antipsychotics: A Medicinal Chemistry Perspective by Giuseppe Felice Mangiatordi, Maria Maddalena Cavalluzzi, Pietro Delre, Giuseppe Lamanna, Maria Cristina Lumuscio, Michele Saviano, Jean-Pierre Majoral, Serge Mignani, Andrea Duranti, Giovanni Lentini

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Revolutionizing Medicinal Chemistry: The Application of Artificial Intelligence (AI) in Early Drug Discovery by Ri Han, Hongryul Yoon, Gahee Kim, Hyundo Lee, Yoonji Lee

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Recent Advances on Quinazoline Derivatives: A Potential Bioactive Scaffold in Medicinal Chemistry by Ram Karan, Pooja Agarwal, Mukty Sinha, Neelima Mahato

“…This paper intended to explore and discover recent therapeutic agents in the area of medicinal chemistry for the treatment of various diseases. …”
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An Overview of the Biological Evaluation of Selected Nitrogen-Containing Heterocycle Medicinal Chemistry Compounds by Oluwakemi Ebenezer, Maryam Amra. Jordaan, Gea Carena, Tommaso Bono, Michael Shapi, Jack A. Tuszynski

“…It explores publications between April 2020 and February 2022 and will benefit researchers in medicinal chemistry and pharmacology. The present work is organized based on the size of the heterocyclic ring.…”
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Editorial to the Special Issue: “Synthesis of Organic Ligands and Their Metal Complexes in Medicinal Chemistry” by Irena Kostova

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SCI-RSC medicinal chemistry sysmposium(3rd:1985: Cambridge, England) Proceedings / by SCI-RSC Medicinal Chemistry Symposium (3rd: 1985 : Cambridge, England), Lambert, R. W.

SCI-RSC medicinal chemistry symposium (2nd: 1983: Cmbridge, England) proceedings / by SCI-RSC Medicinal Chemistry Symposium (2nd : 1983 : Cambridge, England), Emmett, J. C.

Metabolism, pharmacokinetics and toxicity of functional groups : impact of the building blocks of medicinal chemistry in ADMET / by Smith, Dennis A., Royal Society of Chemistry (Great Britain)

30th Annual GP₂A Medicinal Chemistry Conference by Niamh M. O’Boyle, Jean-Jacques Helesbeux, Mary J. Meegan, Astrid Sasse, Elizabeth O’Shaughnessy, Alina Qaisar, Aoife Clancy, Florence McCarthy, Pascal Marchand

Subjects: “…medicinal chemistry…”
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