Are AMPA Receptor Positive Allosteric Modulators Potential Pharmacotherapeutics for Addiction? by Lucas R. Watterson, M. Foster Olive

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The vasorelaxant properties of novel benzodiazepine-like ligands on isolated rat thoracic aorta by Gajić-Bojić Milica, Savić Miroslav

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Experimental GABA A Receptor Agonists and Allosteric Modulators for the Treatment of Focal Epilepsy by Janković SM, Dješević M, Janković SV

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Structural pharmacology of GABAА receptors by Alexey V. Rossokhin, Irina N. Sharonova

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Targeted NMDA Receptor Interventions for Autism: Developmentally Determined Expression of GluN2B and GluN2A-Containing Receptors and Balanced Allosteric Modulatory Approaches by Stephen I. Deutsch, Zachary N. M. Luyo, Jessica A. Burket

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In Silico Prediction and Validation of CB2 Allosteric Binding Sites to Aid the Design of Allosteric Modulators by Jiayi Yuan, Chen Jiang, Junmei Wang, Chih-Jung Chen, Yixuan Hao, Guangyi Zhao, Zhiwei Feng, Xiang-Qun Xie

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A1 Adenosine Receptor Partial Agonists and Allosteric Modulators: Advancing Toward the Clinic? by Fabrizio Vincenzi, Silvia Pasquini, Enrica Battistello, Stefania Merighi, Stefania Gessi, Pier Andrea Borea, Katia Varani

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The structural patterns of the potentiation and the blockade of inhibitory <i>cys</i>-loop receptors through the transmembrane domain by Alexey V. Rossokhin

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Role of mGlu5 in Persistent Forms of Hippocampal Synaptic Plasticity and the Encoding of Spatial Experience by Hardy Hagena, Denise Manahan-Vaughan

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The current agonists and positive allosteric modulators of α7 nAChR for CNS indications in clinical trials by Taoyi Yang, Ting Xiao, Qi Sun, Kewei Wang

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GABAB receptor ligands for the treatment of alcohol use disorder: preclinical and clinical evidence by Roberta eAgabio, Giancarlo eColombo

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Acute Administration of Desformylflustrabromine Relieves Chemically Induced Pain in CD-1 Mice by Loni A. Weggel, Anshul A. Pandya

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Therapeutic potential of α7 nicotinic receptor agonists to regulate neuroinflammation in neurodegenerative diseases by Laura Foucault-Fruchard, Daniel Antier

Subjects: “…α7 nicotinic receptors; cholinergic anti-inflammatory pathway; Alzheimer′s disease; Huntington′s disease; Parkinson′s disease; neuroinflammation; neurodegeneration; positive allosteric modulators…”
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Examining the Effects of (α4)3(β2)2 Nicotinic Acetylcholine Receptor-Selective Positive Allosteric Modulator on Acute Thermal Nociception in Rats by Farah Deba, Kara Ramos, Matthew Vannoy, Kemburli Munoz, Lois S. Akinola, M. Imad Damaj, Ayman K. Hamouda

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The Detrimental Action of Adenosine on Glutamate-Induced Cytotoxicity in PC12 Cells Can Be Shifted towards a Neuroprotective Role through A₁AR Positive Allosteric Modula... by Fabrizio Vincenzi, Silvia Pasquini, Stefania Gessi, Stefania Merighi, Romeo Romagnoli, Pier Andrea Borea, Katia Varani

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Characterization of a novel positive allosteric modulator of the α1A-Adrenergic receptor by Robert S. Papay, Jonathan D. Macdonald, Shaun R. Stauffer, Dianne M. Perez

Subjects: “…Positive allosteric modulator…”
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Positive allosteric regulation of PAC1-R up-regulates<?A3B2 ACK?>PAC1-R and its specific ligand PACAP by Fan Guangchun, Tao Zhengxin, Chen Shang, Zhang Huahua, Yu Rongjie

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Identification of Koumine as a Translocator Protein 18 kDa Positive Allosteric Modulator for the Treatment of Inflammatory and Neuropathic Pain by Bojun Xiong, Bojun Xiong, Guilin Jin, Guilin Jin, Ying Xu, Ying Xu, Wenbing You, Yufei Luo, Menghan Fang, Bing Chen, Huihui Huang, Jian Yang, Jian Yang, Xu Lin, Changxi Yu, Changxi Yu

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Apigenin and Structurally Related Flavonoids Allosterically Potentiate the Function of Human α7-Nicotinic Acetylcholine Receptors Expressed in SH-EP1 Cells by Waheed Shabbir, Keun-Hang Susan Yang, Bassem Sadek, Murat Oz

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De Novo Design of Peptidic Positive Allosteric Modulators Targeting TRPV1 with Analgesic Effects by Lizhen Xu, Heng Zhang, Yunfei Wang, Xiancui Lu, Zhenye Zhao, Cheng Ma, Shilong Yang, Vladimir Yarov‐Yarovoy, Yuhua Tian, Jie Zheng, Fan Yang

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