Bicyclic Basic Merbarone Analogues as Antiproliferative Agents by Andrea Spallarossa, Matteo Lusardi, Chiara Caneva, Aldo Profumo, Camillo Rosano, Marco Ponassi

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Structure–Activity Relationships in NHC–Silver Complexes as Antimicrobial Agents by Luisa Ronga, Mario Varcamonti, Diego Tesauro

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Synthesis and Biological Evaluation of 4β-N-Acetylamino Substituted Podophyllotoxin Derivatives as Novel Anticancer Agents by Jinbao Wei, Jinbao Wei, Jinghong Chen, Peijun Ju, Le Ma, Li Chen, Weidong Ma, Tao Zheng, Guangyi Yang, Yong-Xiang Wang

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Small molecule angiotensin converting enzyme inhibitors: A medicinal chemistry perspective by Wenyue Zheng, Wenyue Zheng, Erkang Tian, Zhen Liu, Changhan Zhou, Pei Yang, Pei Yang, Keyue Tian, Wen Liao, Juan Li, Changyu Ren

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Synthesis and Biochemical Evaluation of 8<i>H</i>-Indeno[1,2-<i>d</i>]thiazole Derivatives as Novel SARS-CoV-2 3CL Protease Inhibitors by Jing Wu, Bo Feng, Li-Xin Gao, Chun Zhang, Jia Li, Da-Jun Xiang, Yi Zang, Wen-Long Wang

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1H-2,3-Dihydroperimidine Derivatives: A New Class of Potent Protein Tyrosine Phosphatase 1B Inhibitors by Wen-Long Wang, Dong-Lin Yang, Li-Xin Gao, Chun-Lan Tang, Wei-Ping Ma, Hui-Hua Ye, Si-Qi Zhang, Ya-Nan Zhao, Hao-Jie Xu, Zhao Hu, Xia Chen, Wen-Hua Fan, Hai-Jun Chen, Jing-Ya Li, Fa-Jun Nan, Jia Li, Bainian Feng

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Defining the hydrophobic interactions that drive competence stimulating peptide (CSP)-ComD binding in Streptococcus pneumoniae by Bimal Koirala, Robert A. Hillman, Erin K. Tiwold, Michael A. Bertucci, Yftah Tal-Gan

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Identification of Bioactive Compounds from Marine Natural Products and Exploration of Structure-Activity Relationships (SAR) by Mojdeh Dinarvand, Malcolm Spain

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Antimicrobial Peptides for Therapeutic Applications: A Review by Tsogbadrakh Mishig-Ochir, Ji-Hun Kim, Min-Duk Seo, Hyung-Sik Won, Bong-Jin Lee

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Semi-Synthesis of Harringtonolide Derivatives and Their Antiproliferative Activity by Xiutao Wu, Lijie Gong, Chen Chen, Ye Tao, Wuxi Zhou, Lingyi Kong, Jianguang Luo

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Comparative Antibacterial Activities of Some Monosaccharide and Disaccharide Benzoates by Mohammed M. Matin, Mohammed H. Bhuiyan, Mohammed Manir Hossain, Mohammad Harun Or Roshid

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Synthesis and Antimicrobial Evaluation of Novel Pyrazolopyrimidines Incorporated with Mono- and Diphenylsulfonyl Groups by Amani M. R. Alsaedi, Thoraya. A. Farghaly, Mohamed R. Shaaban

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Upregulation of p53 through induction of MDM2 degradation: improved potency through the introduction of an alkylketone sidechain on the anthraquinone core by Ravi Tripathi, Abiodun Anifowose, Wen Lu, Xiaoxiao Yang, Binghe Wang

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Synthesis, Insecticidal, Fungicidal Activities and Structure–Activity Relationships of Tschimganin Analogs by Yueting Zhou, Chunjuan Wang, Fang Xin, Xiaoqiang Han, Jie Zhang, Ke Sun

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Synthesis and biological evaluation of C-4 substituted phenoxazine-bearing hydroxamic acids with potent class II histone deacetylase inhibitory activities by Jung-Chun Chu, Hui-Ju Tseng, Sung-Bau Lee, Kai-Cheng Hsu, Ling-Wei Hsin, Ru-Hao Liang, Tony Eight Lin, Nain-Chu Gao, Liang-Chieh Chen, Wan-Hsun Lu, Andrew H.-J Wang, Wei-Jan Huang

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Design, Synthesis and Biological Evaluation of 1,4-Benzenesulfonamide Derivatives as Glyoxalase I Inhibitors by Audat SA, Al-Balas QA, Al-Oudat BA, Athamneh MJ, Bryant-Friedrich A

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A Comprehensive Overview of the Antibiotics Approved in the Last Two Decades: Retrospects and Prospects by Zhenfeng Shi, Jie Zhang, Lei Tian, Liang Xin, Chengyuan Liang, Xiaodong Ren, Min Li

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Design, synthesis, and biological evaluation of novel N 4 -substituted sulfonamides: acetamides derivatives as dihydrofolate reductase (DHFR) inhibitors by Essam M. Hussein, Munirah M. Al-Rooqi, Shimaa M. Abd El-Galil, Saleh A. Ahmed

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Structure–Activity Relationship Analysis of Flavonoids and Its Inhibitory Activity Against BACE1 Enzyme Toward a Better Therapy for Alzheimer’s Disease by Nur Intan Saidaah Mohamed Yusof, Zafirah Liyana Abdullah, Norodiyah Othman, Norodiyah Othman, Fazlin Mohd Fauzi, Fazlin Mohd Fauzi

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Structure-activity correlations for peptaibols obtained from clade Longibrachiatum of Trichoderma: A combined experimental and computational approach by Dóra Balázs, Tamás Marik, András Szekeres, Csaba Vágvölgyi, László Kredics, Chetna Tyagi

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