Thienopyrimidine: A Promising Scaffold to Access Anti-Infective Agents by Prisca Lagardère, Cyril Fersing, Nicolas Masurier, Vincent Lisowski

Subjects: “…thienopyrimidine…”
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In Vitro Anticancer Activity Screening of Novel Fused Thiophene Derivatives as VEGFR-2/AKT Dual Inhibitors and Apoptosis Inducers by Rana M. Abdelnaby, Afaf A. El-Malah, Rasha R. FakhrEldeen, Marwa M. Saeed, Rania I. Nadeem, Nancy S. Younis, Hanaa M. Abdel-Rahman, Nehad M. El-Dydamony

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Design, Synthesis, and Biological Evaluation of Novel Thienopyrimidine Derivatives as PI3Kα Inhibitors by Lide Yu, Qinqin Wang, Caolin Wang, Binliang Zhang, Zunhua Yang, Yuanying Fang, Wufu Zhu, Pengwu Zheng

Subjects: “…Thienopyrimidine…”
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4-Substituted Thieno[3,2-<i>d</i>]pyrimidines as Dual-Stage Antiplasmodial Derivatives by Prisca Lagardère, Romain Mustière, Nadia Amanzougaghene, Sébastien Hutter, Jean-François Franetich, Nadine Azas, Patrice Vanelle, Pierre Verhaeghe, Nicolas Primas, Dominique Mazier, Nicolas Masurier, Vincent Lisowski

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Antimicrobial Evaluation of Sulfonamides after Coupling with Thienopyrimidine Coplanar Structure by Elshaymaa I. Elmongy, Wejdan S. Alanazi, Alhanouf I. Aldawsari, Asma A. Alfaouri, Reem Binsuwaidan

Subjects: “…thienopyrimidine–sulfonamide hybrids…”
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Synthesis and Cytotoxicity Assay of Aniline Substituted Thienopyrimidines for Anti-Colorectal Cancer Activity by Mahalakshmi Suresha Biradar, Shachindra L. Nargund, Shankar Thapa

Subjects: “…Thienopyrimidine…”
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Combined 3D-QSAR and Molecular Docking Analysis of Thienopyrimidine Derivatives as Staphylococcus aureus Inhibitors by Mebarka Ouassaf, Salah Belaidi, Saida Khamouli, Houmam Belaidi, Samir Chtita

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Design, synthesis, biological evaluation, and bio-computational modeling of imidazo, thieno, pyrimidopyrimidine, pyrimidodiazepene, and motifs as antimicrobial agents by El-Ahwany Maged F., Assy Mohamed G., Sherif Mohamed H., Soliman Mohamed R., Titi Abderrahim, Touzani Rachid, El-Gendey Marwa S., Shehab Wesam S., Abdellattif Magda H.

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Starch Nanoparticles for Enhancement of Oral Bioavailability of a Newly Synthesized Thienopyrimidine Derivative with Anti-Proliferative Activity Against Pancreatic Cancer by Gardouh AR, Srag El-Din AS, Salem MSH, Moustafa Y, Gad S

Subjects: “…thienopyrimidine derivative…”
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Synthesis of Novel Analogs of Thieno[2,3-<i>d</i>] Pyrimidin-4(3<i>H</i>)-ones as Selective Inhibitors of Cancer Cell Growth by Sheng Zhang, Feize Liu, Xueling Hou, Jianguo Cao, Xiling Dai, Junjie Yu, Guozheng Huang

Subjects: “…thienopyrimidine…”
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Synthesis and biological evaluation of novel thienopyrimidine derivatives as diacylglycerol acyltransferase 1 (DGAT-1) inhibitors by Dong Jin Hong, Seung Hyun Jung, Jisook Kim, Danbee Jung, Young Gil Ahn, Kwee Hyun Suh, Kyung Hoon Min

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Fragment merging approach for design, synthesis, and biological assessment of urea/acetyl hydrazide clubbed thienopyrimidine derivatives as GSK-3β inhibitors by Joseph S. Saleh, Soha R. Abd El Hadi, Hany S. Ibrahim, Eman Z. Elrazaz, Khaled A. M. Abouzid

Subjects: “…Thienopyrimidine…”
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Synthesis, molecular modelling and biological evaluation of new 4-aminothiophene and thienopyrimidine compounds by Aisha Hossan, Mansoor Alsahag, Ali Alisaac, Majid A. Bamaga, Adel I. Alalawy, Nashwa M. El-Metwaly

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Click chemistry based synthesis, cytotoxic activity and molecular docking of novel triazole-thienopyrimidine hybrid glycosides targeting EGFR by Reham R. Khattab, Asma K. Alshamari, Allam A. Hassan, Hussein H. Elganzory, Wael A. El-Sayed, Hanem M. Awad, Eman S. Nossier, Nasser A. Hassan

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Pyridine-Based Heterocycles. Synthesis of New Pyrido [4',3':4,5]thieno[2,3-d]pyrimidines and Related Heterocycles by Hussein El-Kashef, Abdel-Rahman Farghaly, Ahmed Al-Hazmi, Thierry Terme, Patrice Vanelle

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In Silico Evaluation of a Promising Key Intermediate Thieno [2,3-d] Pyrimidine Derivative with Expected JAK2 Kinase Inhibitory Activity by Elshaymaa I. Elmongy, Hanan Ali Henidi

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Synthesis of Some Thienopyrimidine Derivatives by Hassan M. Al-Hazimi, Hanan A. S. Al-Blowy, Fatma E. M. El-Baih

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Synthesis and Pharmacological Activities of Some New Triazolo- and Tetrazolopyrimidine Derivatives by Saleh A. Bahashwan, Ahmed A. Fayed, Abd El-Galil E. Amr, Eman M. Flefel, Atef Kalmouch

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In-Silico Screening of Novel Synthesized Thienopyrimidines Targeting Fms Related Receptor Tyrosine Kinase-3 and Their In-Vitro Biological Evaluation by Elshaymaa I. Elmongy, Najla Altwaijry, Nashwah G. M. Attallah, Manal Mubarak AlKahtani, Hanan Ali Henidi

Subjects: “…thienopyrimidines…”
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Design, Cytotoxicity and Antiproliferative Activity of 4-Amino-5-methyl-thieno[2,3-d]pyrimidine-6-carboxylates against MFC-7 and MDA-MB-231 Breast Cancer Cell Lines by Anelia Mavrova, Stephan Dimov, Inna Sulikovska, Denitsa Yancheva, Ivan Iliev, Iana Tsoneva, Galya Staneva, Biliana Nikolova

Subjects: “…4-amino-thienopyrimidines…”
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