Synthesis of Galectin Inhibitors by Regioselective 3′-<i>O</i>-Sulfation of Vanillin Lactosides Obtained under Phase Transfer Catalysis

Vanillin-based lactoside derivatives were synthetized using phase-transfer catalyzed reactions from per-<i>O</i>-acetylated lactosyl bromide. The aldehyde group of the vanillin moiety was then modified to generate a series of related analogs having variable functionalities in the <i&g...

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Bibliographic Details
Main Authors: Karima Belkhadem, Yihong Cao, René Roy
Format: Article
Language:English
Published: MDPI AG 2020-12-01
Series:Molecules
Subjects:
Online Access:https://www.mdpi.com/1420-3049/26/1/115